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Example1
Example2
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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
8 JAK1 related diseases
hsa05140
Leishmaniasis
hsa05145
Toxoplasmosis
hsa05152
Tuberculosis
hsa05160
Hepatitis C
hsa05162
Measles
hsa05164
Influenza A
hsa05168
Herpes simplex infection
hsa05169
Epstein-Barr virus infection
Summary of query kinase
Query kinase
JAK1 (
P23458
)
Kinase group
TK
Number of conformation types
1
Number of structural templates
2 (
Total 129 inhibitors
)
Number of JAK1 related diseases
8 (
hsa05140
hsa05145
hsa05152
hsa05160
hsa05162
hsa05164
hsa05168
hsa05169
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
B
2
3EYHA_IZA
(JAK1)
TK
Pyridone 6
I
21
19
54
B
3EYHA_IZA
(JAK1)
TK
Pyridone 6
I
21
19
54
21
19
54
B
3EYGA_MI1
(JAK1)
TK
CP690550
I
8
23
31
8
23
31