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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
HIPK3 (
Q9H422
)
Kinase group
CMGC
Number of conformation types
0
Number of structural templates
29 (
Total 39 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
17
2JAMA_J60
(CAMK1G)
CMGC
SU11652
I
50
65
32
A
2JAMA_J60
(CAMK1G)
CMGC
SU11652
I
50
65
32
50
65
32
A
1AQ1A_STU
(CDK2)
CMGC
staurosporine
I
195
76
118
195
76
118
A
1Q3DA_STU
(GSK3B)
CMGC
staurosporine
I
115
71
61
115
71
61
A
2VTTA_LZD
(CDK2)
CMGC
pyrazole dia...
I
158
42
111
158
42
111
A
1PKDA_UCN
(CDK2)
CMGC
UCN 02
I
195
67
118
195
67
118
A
2O0UA_C0M
(MAPK10)
CMGC
ZINC00799686
I
21
8
23
21
8
23
A
3MVLA_38P
(MAPK14)
CMGC
38P
I
50
308
44
50
308
44
A
3BLRA_CPB
(CDK9)
CMGC
BIIVYFLTOXDA...
I
48
17
41
48
17
41
A
2IW6A_QQ2
(CDK2)
CMGC
2iw6
I
112
209
86
112
209
86
A
2ZB1A_GK4
(MAPK14)
CMGC
biphenyl ami...
II
55
57
54
55
57
54
A
1R78A_FMD
(CDK2)
CMGC
4-alkynyl ox...
I
127
24
97
127
24
97
A
3E92A_G6A
(MAPK14)
CMGC
3e92
I
56
59
55
56
59
55
A
2I0EA_PDS
(PRKCB)
CMGC
bisindolylma...
I
41
141
45
41
141
45
A
3IPHA_G11
(MAPK14)
CMGC
HMS3303K05
I
57
108
55
57
108
55
A
2OW3A_BIM
(GSK3B)
CMGC
LY_333531
I
62
139
51
62
139
51
A
3L8XA_N4D
(MAPK14)
CMGC
3cg2
I
91
104
65
91
104
65
A
3IW4A_LW4
(PRKCA)
CMGC
Sotrastaurin
I
52
119
49
52
119
49
B
12
1WVYA_STU
(DAPK1)
CMGC
staurosporine
I
83
23
55
B
1WVYA_STU
(DAPK1)
CMGC
staurosporine
I
83
23
55
83
23
55
B
2PE2A_464
(PDPK1)
CMGC
Indolinone b...
I
134
156
104
134
156
104
B
1OKYA_STU
(PDPK1)
CMGC
staurosporine
I
179
67
109
179
67
109
B
1OKZA_UCN
(PDPK1)
CMGC
UCN 02
I
179
60
109
179
60
109
B
1UU3A_LY4
(PDPK1)
CMGC
Ruboxistaurin
I
71
117
57
71
117
57
B
3ORZA_BI4
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU7A_BI2
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65
B
3OTUA_BI4
(PDPK1)
CMGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU8A_BI1
(PDPK1)
CMGC
bisindolylma...
I
83
189
65
83
189
65
B
1H07A_MFP
(CDK2)
CMGC
AC1NAKJQ
I
90
241
80
90
241
80
B
1UU9A_BI3
(PDPK1)
CMGC
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
1UVRA_BI8
(PDPK1)
CMGC
Ro 31-7549
I
82
181
65
82
181
65