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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
PCTK2 (
Q00537
)
Kinase group
CMGC
Number of conformation types
0
Number of structural templates
22 (
Total 37 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
12
2VTTA_LZD
(CDK2)
CMGC
pyrazole dia...
I
158
42
111
A
2VTTA_LZD
(CDK2)
CMGC
pyrazole dia...
I
158
42
111
158
42
111
A
1PKDA_UCN
(CDK2)
CMGC
UCN 02
I
195
67
118
195
67
118
A
1Q3DA_STU
(GSK3B)
CMGC
staurosporine
I
115
71
61
115
71
61
A
1AQ1A_STU
(CDK2)
CMGC
staurosporine
I
195
76
118
195
76
118
A
1NVQA_UCN
(CHEK1)
CMGC
UCN 02
I
179
65
79
179
65
79
A
1NVRA_STU
(CHEK1)
CMGC
staurosporine
I
179
71
79
179
71
79
A
3CKXA_STU
(STK24)
CMGC
staurosporine
I
176
104
141
176
104
141
A
3BLRA_CPB
(CDK9)
CMGC
BIIVYFLTOXDA...
I
48
17
41
48
17
41
A
1R0EA_DFN
(GSK3B)
CMGC
HMS3401D14
I
17
17
17
17
17
17
A
2VTQA_LZA
(CDK2)
CMGC
pyrazole dia...
I
36
25
31
36
25
31
A
2VU3A_LZE
(CDK2)
CMGC
AT7519
I
35
22
29
35
22
29
A
2WIHA_P48
(CDK2)
CMGC
VX_680
I
111
425
105
111
425
105
B
9
2PE2A_464
(PDPK1)
CMGC
Indolinone b...
I
134
156
104
B
2PE2A_464
(PDPK1)
CMGC
Indolinone b...
I
134
156
104
134
156
104
B
2WKMA_PFY
(MET)
CMGC
PHA-665752
I
38
34
98
38
34
98
B
3MIYA_B49
(ITK)
CMGC
Sunitinib
I
70
74
110
70
74
110
B
1OKZA_UCN
(PDPK1)
CMGC
UCN 02
I
179
60
109
179
60
109
B
3BKBA_STU
(FES)
CMGC
staurosporine
I
131
107
138
131
107
138
B
3CBLA_STU
(FES)
CMGC
staurosporine
I
131
107
138
131
107
138
B
3CD3A_STU
(FES)
CMGC
staurosporine
I
131
107
138
131
107
138
B
1OKYA_STU
(PDPK1)
CMGC
staurosporine
I
179
67
109
179
67
109
B
2FVDA_LIA
(CDK2)
CMGC
[4-Amino-2-[...
I
39
16
29
39
16
29
D
1
1R0PA_KSA
(MET)
CMGC
k-252a
I
28
79
64
D
1R0PA_KSA
(MET)
CMGC
k-252a
I
28
79
64
28
79
64