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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
LY4
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
PIM1 (PDB code: 2J2I)
[PDB]
[PDBsum]
Inhibitor
Ruboxistaurin (HET code: LY4)
[PDB]
Summary of KIF 2J2IB_LY4
(PIM1, PDB code:
2J2I
, chain B)
Number of family interactions
347
Number of family kinase
35 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
89 (3 are AKT3 inhibitors)
Involved diseases
36 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
AKT3 and 3 inhibitors