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Example2
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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
WTI
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
CHEK2 (PDB code: 2WTI)
[PDB]
[PDBsum]
Inhibitor
WTI (HET code: WTI)
[PDB]
Summary of KIF 2WTIA_WTI
(CHEK2, PDB code:
2WTI
, chain A)
Number of family interactions
28
Number of family kinase
4 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
20 (14 are CHEK2 inhibitors)
Involved diseases
6 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
CHEK2 and 14 inhibitors