Protein Surface  Ribbon
Inhibitor LWH
  ATP Location
Pocket ATP NLP HAP CLP SP
Selected template
Kinase CHEK2 (PDB code: 2XM9) [PDB] [PDBsum]
Inhibitor 4-(1h-Pyrazol-5-Yl)-2-{4-[(3s)-Pyrrolidin-3-Ylamino]quinazolin-2-Yl}phenol (HET code: LWH) [PDB]
 
Summary of KIF 2XM9A_LWH (CHEK2, PDB code: 2XM9, chain A)
Number of family interactions 42
Number of family kinase 5 (sequence conservation) (profiling results)
Number of family inhibitors 34 (21 are CHEK2 inhibitors)
Involved diseases 17 (show)
Number of family anchors  
All kinase-inhibitor interactions in this family  CHEK2 and 21 inhibitors