Protein Surface  Ribbon
Inhibitor R78
  ATP Location
Pocket ATP NLP HAP CLP SP
Selected template
Kinase PLK1 (PDB code: 2RKU) [PDB] [PDBsum]
Inhibitor BI 2536 (HET code: R78) [PDB]
 
Summary of KIF 2RKUA_R78 (PLK1, PDB code: 2RKU, chain A)
Number of family interactions 103
Number of family kinase 37 (sequence conservation) (profiling results)
Number of family inhibitors 59 (1 are GRK7 inhibitors)
Involved diseases 35 (show)
Number of family anchors  
All kinase-inhibitor interactions in this family  GRK7 and 1 inhibitors