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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
5B3
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
JAK2 (PDB code: 3E64)
[PDB]
[PDBsum]
Inhibitor
3e64 (HET code: 5B3)
[PDB]
Summary of KIF 3E64A_5B3
(JAK2, PDB code:
3E64
, chain A)
Number of family interactions
11
Number of family kinase
3 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
10 (9 are JAK2 inhibitors)
Involved diseases
20 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
JAK2 and 9 inhibitors