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KIDFamMap
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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
NVB
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
JAK2 (PDB code: 3LPB)
[PDB]
[PDBsum]
Inhibitor
Anilinopyrazole deriv. 1j (HET code: NVB)
[PDB]
Summary of KIF 3LPBA_NVB
(JAK2, PDB code:
3LPB
, chain A)
Number of family interactions
15
Number of family kinase
6 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
8 (4 are JAK2 inhibitors)
Involved diseases
19 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
JAK2 and 4 inhibitors