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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
SX8
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
MET (PDB code: 3DKG)
[PDB]
[PDBsum]
Inhibitor
1-{[6-(pyridin-3-yl)[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-3-yl]methyl}-1H-benzimidazole (HET code: SX8)
[PDB]
Summary of KIF 3DKGA_SX8
(MET, PDB code:
3DKG
, chain A)
Number of family interactions
9
Number of family kinase
3 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
5 (3 are MET inhibitors)
Involved diseases
11 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
MET and 3 inhibitors