Summary of query kinase
Query kinase CSNK1G1 (Q9HCP0)
Kinase group CK1
Number of inhibitors 29
Index Target Inhibitor Inhibitor 2D Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) POC Source Link
0 CSNK1G1 CHEMBL511410 BD50259563 n/a 160 n/a n/a n/a BindingDB BindingDB
1 CSNK1G1 CHEMBL466496 BD50259376 n/a 250 n/a n/a n/a BindingDB BindingDB
2 CSNK1G1 CHEMBL519113 BD50259637 n/a 4900 n/a n/a n/a BindingDB BindingDB
3 CSNK1G1 CHEMBL467079 BD50259532 n/a 520 n/a n/a n/a BindingDB BindingDB
4 CSNK1G1 CHEMBL1087650 BD50311985 n/a 9510 n/a n/a n/a BindingDB BindingDB
5 CSNK1G1 cid_10138259 BD00031095 n/a n/a 1000 n/a n/a BindingDB BindingDB
6 CSNK1G1 AST_487 AST_487 n/a n/a 1000 n/a n/a NB2011DRx NB2011DRx
7 CSNK1G1 SU_14813 SU_14813 n/a n/a 1000 n/a n/a NB2008 NB2008
8 CSNK1G1 SU_14813 SU_14813 n/a n/a 1000 n/a n/a NB2011DRx NB2011DRx
9 CSNK1G1 JNJ-7706621 BD00006866 n/a n/a 1200 n/a n/a BindingDB BindingDB
10 CSNK1G1 Flavopiridol Flavopiridol n/a n/a 1200 n/a n/a NB2011DRx NB2011DRx
11 CSNK1G1 JNJ_7706621 JNJ_7706621 n/a n/a 1200 n/a n/a NB2008 NB2008
12 CSNK1G1 KW_2449 KW_2449 n/a n/a 1200 n/a n/a NB2011DRx NB2011DRx
13 CSNK1G1 (R)-Roscovitine BD00007533 n/a n/a 3300 n/a n/a BindingDB BindingDB
14 CSNK1G1 Staurosporine Staurosporine n/a n/a 3500 n/a n/a NB2011DRx NB2011DRx
15 CSNK1G1 SP600125 BD00016018 n/a n/a 3700 n/a n/a BindingDB BindingDB
16 CSNK1G1 PP_242 PP_242 n/a n/a 3900 n/a n/a NB2011DRx NB2011DRx
17 CSNK1G1 BI_2536 BI_2536 n/a n/a 4500 n/a n/a NB2011DRx NB2011DRx
18 CSNK1G1 A_674563 A_674563 n/a n/a 530 n/a n/a NB2011DRx NB2011DRx
19 CSNK1G1 TG_100_115 TG_100_115 n/a n/a 5700 n/a n/a NB2011DRx NB2011DRx
20 CSNK1G1 CHEMBL526901 BD50273635 n/a n/a 59 n/a n/a BindingDB BindingDB
21 CSNK1G1 SU11248 BD00004814 n/a n/a 930 n/a n/a BindingDB BindingDB
22 CSNK1G1 Sunitinib Sunitinib n/a n/a 930 n/a n/a NB2008 NB2008
23 CSNK1G1 Sunitinib Sunitinib n/a n/a 930 n/a n/a NB2011DRx NB2011DRx
24 CSNK1G1 CAS212779_48_1 CAS212779_48_1 n/a n/a n/a n/a 16.03 NB2011RBC NB2011RBC
25 CSNK1G1 CAS212844_53_6 CAS212844_53_6 n/a n/a n/a n/a 28.02 NB2011RBC NB2011RBC
26 CSNK1G1 CAS220792_57_4 CAS220792_57_4 n/a n/a n/a n/a 26.43 NB2011RBC NB2011RBC
27 CSNK1G1 CAS443798_55_8 CAS443798_55_8 n/a n/a n/a n/a 16.71 NB2011RBC NB2011RBC
28 CSNK1G1 OLP OLP n/a n/a n/a n/a n/a PDB PDB