Summary of query kinase
Query kinase DAPK3 (O43293)
Kinase group CAMK
Number of inhibitors 74
Index Target Inhibitor Inhibitor 2D Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) POC Source Link
0 DAPK3 CHEMBL1091041 BD50314672 n/a 148.4 n/a n/a n/a BindingDB BindingDB
1 DAPK3 CHEMBL1091042 BD50314673 n/a 157 n/a n/a n/a BindingDB BindingDB
2 DAPK3 CHEMBL1230165 BD50335638 n/a 17 n/a n/a n/a BindingDB BindingDB
3 DAPK3 CHEMBL1091784 BD50314664 n/a 227.1 n/a n/a n/a BindingDB BindingDB
4 DAPK3 CHEMBL1091785 BD50314665 n/a 278.5 n/a n/a n/a BindingDB BindingDB
5 DAPK3 CHEMBL1091766 BD50314670 n/a 278.5 n/a n/a n/a BindingDB BindingDB
6 DAPK3 CHEMBL1092139 BD50314671 n/a 291.2 n/a n/a n/a BindingDB BindingDB
7 DAPK3 CHEMBL1091764 BD50314668 n/a 346.1 n/a n/a n/a BindingDB BindingDB
8 DAPK3 CHEMBL1091765 BD50314669 n/a 359.6 n/a n/a n/a BindingDB BindingDB
9 DAPK3 CHEMBL1094004 BD50314674 n/a 395.3 n/a n/a n/a BindingDB BindingDB
10 DAPK3 CHEMBL590109 BD50305006 n/a 4300 n/a n/a n/a BindingDB BindingDB
11 DAPK3 CHEMBL1091787 BD50314667 n/a 529.5 n/a n/a n/a BindingDB BindingDB
12 DAPK3 CHEMBL1094005 BD50314675 n/a 533.5 n/a n/a n/a BindingDB BindingDB
13 DAPK3 CHEMBL579387 BD50314663 n/a 583 n/a n/a n/a BindingDB BindingDB
14 DAPK3 CHEMBL1091786 BD50314666 n/a 713.7 n/a n/a n/a BindingDB BindingDB
15 DAPK3 Staurosporine BD00002579 n/a n/a 1 n/a n/a BindingDB BindingDB
16 DAPK3 CHEMBL162 BD50059889 n/a n/a 1 n/a n/a BindingDB BindingDB
17 DAPK3 Staurosporine Staurosporine n/a n/a 1 n/a n/a NB2008 NB2008
18 DAPK3 Staurosporine Staurosporine n/a n/a 1 n/a n/a NB2011DRx NB2011DRx
19 DAPK3 TG_101348 TG_101348 n/a n/a 1.2 n/a n/a NB2011DRx NB2011DRx
20 DAPK3 cid_451705 BD00031096 n/a n/a 1000 n/a n/a BindingDB BindingDB
21 DAPK3 A_674563 A_674563 n/a n/a 1200 n/a n/a NB2011DRx NB2011DRx
22 DAPK3 GSK_1838705A GSK_1838705A n/a n/a 1200 n/a n/a NB2011DRx NB2011DRx
23 DAPK3 R406 R406 n/a n/a 13 n/a n/a NB2011DRx NB2011DRx
24 DAPK3 BI_2536 BI_2536 n/a n/a 130 n/a n/a NB2011DRx NB2011DRx
25 DAPK3 LY333531 BD00017055 n/a n/a 1300 n/a n/a BindingDB BindingDB
26 DAPK3 cid_10138259 BD00031095 n/a n/a 170 n/a n/a BindingDB BindingDB
27 DAPK3 SU_14813 SU_14813 n/a n/a 170 n/a n/a NB2008 NB2008
28 DAPK3 SU_14813 SU_14813 n/a n/a 170 n/a n/a NB2011DRx NB2011DRx
29 DAPK3 CHEBI:668343 BD50298227 n/a n/a 1800 n/a n/a BindingDB BindingDB
30 DAPK3 CHEMBL608533 BD50326053 n/a n/a 1800 n/a n/a BindingDB BindingDB
31 DAPK3 GDC_0941 GDC_0941 n/a n/a 1800 n/a n/a NB2011DRx NB2011DRx
32 DAPK3 PKC_412 PKC_412 n/a n/a 1800 n/a n/a NB2008 NB2008
33 DAPK3 PKC_412 PKC_412 n/a n/a 1800 n/a n/a NB2011DRx NB2011DRx
34 DAPK3 VX-680 BD00013534 n/a n/a 190 n/a n/a BindingDB BindingDB
35 DAPK3 CHEMBL522892 BD50265677 n/a n/a 2100 n/a n/a BindingDB BindingDB
36 DAPK3 BIBF_1120der BIBF_1120der n/a n/a 2100 n/a n/a NB2011DRx NB2011DRx
37 DAPK3 SU11248 BD00004814 n/a n/a 22 n/a n/a BindingDB BindingDB
38 DAPK3 Sunitinib Sunitinib n/a n/a 22 n/a n/a NB2008 NB2008
39 DAPK3 Sunitinib Sunitinib n/a n/a 22 n/a n/a NB2011DRx NB2011DRx
40 DAPK3 TAE_684 TAE_684 n/a n/a 2200 n/a n/a NB2011DRx NB2011DRx
41 DAPK3 cid_11409972 BD00031085 n/a n/a 2500 n/a n/a BindingDB BindingDB
42 DAPK3 CHEBI:259924 BD50119072 n/a n/a 2600 n/a n/a BindingDB BindingDB
43 DAPK3 KW_2449 KW_2449 n/a n/a 310 n/a n/a NB2011DRx NB2011DRx
44 DAPK3 EXEL_2880 EXEL_2880 n/a n/a 3100 n/a n/a NB2011DRx NB2011DRx
45 DAPK3 AST_487 AST_487 n/a n/a 3200 n/a n/a NB2008 NB2008
46 DAPK3 AST_487 AST_487 n/a n/a 3200 n/a n/a NB2011DRx NB2011DRx
47 DAPK3 PP_242 PP_242 n/a n/a 41 n/a n/a NB2011DRx NB2011DRx
48 DAPK3 SP600125 BD00016018 n/a n/a 410 n/a n/a BindingDB BindingDB
49 DAPK3 cid_6445562 BD00031090 n/a n/a 4100 n/a n/a BindingDB BindingDB
50 DAPK3 JNJ_28312141 JNJ_28312141 n/a n/a 4700 n/a n/a NB2011DRx NB2011DRx
51 DAPK3 JNJ-7706621 BD00006866 n/a n/a 5200 n/a n/a BindingDB BindingDB
52 DAPK3 GSK_461364A GSK_461364A n/a n/a 5500 n/a n/a NB2011DRx NB2011DRx
53 DAPK3 GSK_690693 GSK_690693 n/a n/a 560 n/a n/a NB2011DRx NB2011DRx
54 DAPK3 Iressa BD00005447 n/a n/a 5700 n/a n/a BindingDB BindingDB
55 DAPK3 Gefitinib Gefitinib n/a n/a 5700 n/a n/a NB2008 NB2008
56 DAPK3 Gefitinib Gefitinib n/a n/a 5700 n/a n/a NB2011DRx NB2011DRx
57 DAPK3 Erlotinib Erlotinib n/a n/a 6000 n/a n/a NB2011DRx NB2011DRx
58 DAPK3 LY_333531 LY_333531 n/a n/a 8000 n/a n/a NB2011DRx NB2011DRx
59 DAPK3 CHEMBL603469 BD50308060 n/a n/a 82 n/a n/a BindingDB BindingDB
60 DAPK3 CEP_701 CEP_701 n/a n/a 82 n/a n/a NB2011DRx NB2011DRx
61 DAPK3 pyridofuropyrimidine derivative, 2 BD00025045 n/a n/a 840 n/a n/a BindingDB BindingDB
62 DAPK3 PI_103 PI_103 n/a n/a 840 n/a n/a NB2008 NB2008
63 DAPK3 PI_103 PI_103 n/a n/a 840 n/a n/a NB2011DRx NB2011DRx
64 DAPK3 INCB18424 INCB18424 n/a n/a 89 n/a n/a NB2011DRx NB2011DRx
65 DAPK3 VX_680 VX_680 n/a n/a 9900 n/a n/a NB2011DRx NB2011DRx
66 DAPK3 4RB 4RB n/a n/a n/a n/a n/a PDB PDB
67 DAPK3 7CP 7CP n/a n/a n/a n/a n/a PDB PDB
68 DAPK3 CAS135897_06_2 CAS135897_06_2 n/a n/a n/a n/a 24.58 NB2011RBC NB2011RBC
69 DAPK3 CAS244148_46_7 CAS244148_46_7 n/a n/a n/a n/a 29.61 NB2011RBC NB2011RBC
70 DAPK3 CAS457081_03_7 CAS457081_03_7 n/a n/a n/a n/a 2.18 NB2011RBC NB2011RBC
71 DAPK3 CAS62996_74_1 CAS62996_74_1 n/a n/a n/a n/a 1.91 NB2011RBC NB2011RBC
72 DAPK3 CAS97161_97_2 CAS97161_97_2 n/a n/a n/a n/a 27.17 NB2011RBC NB2011RBC
73 DAPK3 IZA IZA n/a n/a n/a n/a n/a PDB PDB