Summary of query kinase
Query kinase INSR (P06213)
Kinase group TK
Number of inhibitors 322
Index Target Inhibitor Inhibitor 2D Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) POC Source Link
0 INSR CHEMBL514873 BD50265869 n/a 0.4 n/a n/a n/a BindingDB BindingDB
1 INSR CHEMBL515519 BD50265888 n/a 0.8 n/a n/a n/a BindingDB BindingDB
2 INSR CHEMBL1642137 BD50333563 n/a 1000 n/a n/a n/a BindingDB BindingDB
3 INSR CHEMBL381738 BD50181675 9000 10100 n/a n/a n/a BindingDB BindingDB
4 INSR CHEMBL601719 BD50306682 n/a 102 n/a n/a n/a BindingDB BindingDB
5 INSR CHEMBL1076472 BD50311934 n/a 1087 n/a n/a n/a BindingDB BindingDB
6 INSR CHEMBL1076202 BD50311913 n/a 1092 n/a n/a n/a BindingDB BindingDB
7 INSR CHEMBL1644800 BD50334086 n/a 11 n/a n/a n/a BindingDB BindingDB
8 INSR CHEMBL457886 BD50274749 n/a 110 n/a n/a n/a BindingDB BindingDB
9 INSR CHEMBL209148 BD50186460 n/a 1100 n/a n/a n/a BindingDB BindingDB
10 INSR CHEMBL493008 BD50257916 n/a 1100 n/a n/a n/a BindingDB BindingDB
11 INSR CHEMBL1822525 BD50353046 n/a 1137 n/a n/a n/a BindingDB BindingDB
12 INSR CHEMBL1076468 BD50311930 n/a 1141 n/a n/a n/a BindingDB BindingDB
13 INSR CHEMBL1644810 BD50334083 n/a 1150 n/a n/a n/a BindingDB BindingDB
14 INSR CHEMBL1822526 BD50353047 n/a 1171 n/a n/a n/a BindingDB BindingDB
15 INSR CHEMBL485202 BD50274702 n/a 120 n/a n/a n/a BindingDB BindingDB
16 INSR CHEMBL499219 BD50257752 n/a 1200 n/a n/a n/a BindingDB BindingDB
17 INSR CHEMBL1642149 BD50333575 n/a 1200 n/a n/a n/a BindingDB BindingDB
18 INSR CHEMBL1076198 BD50311909 n/a 1221 n/a n/a n/a BindingDB BindingDB
19 INSR CHEMBL1087128 BD50311898 n/a 1224 n/a n/a n/a BindingDB BindingDB
20 INSR CHEMBL1822515 BD50353052 n/a 123 n/a n/a n/a BindingDB BindingDB
21 INSR CHEMBL485555 BD50274470 n/a 125 n/a n/a n/a BindingDB BindingDB
22 INSR CHEMBL1630111 BD50332484 n/a 1300 n/a n/a n/a BindingDB BindingDB
23 INSR CHEMBL1076203 BD50311915 n/a 1365 n/a n/a n/a BindingDB BindingDB
24 INSR CHEMBL1642258 BD50334593 n/a 1380 n/a n/a n/a BindingDB BindingDB
25 INSR CHEMBL485564 BD50274205 n/a 140 n/a n/a n/a BindingDB BindingDB
26 INSR CHEMBL1083527 BD50313651 n/a 140 n/a n/a n/a BindingDB BindingDB
27 INSR CHEMBL1630117 BD50332490 n/a 1400 n/a n/a n/a BindingDB BindingDB
28 INSR CHEMBL1642140 BD50333566 n/a 1400 n/a n/a n/a BindingDB BindingDB
29 INSR CHEMBL1796254 BD50347053 n/a 1400 n/a n/a n/a BindingDB BindingDB
30 INSR CHEMBL1076477 BD50311939 n/a 1435 n/a n/a n/a BindingDB BindingDB
31 INSR CHEMBL1076473 BD50311935 n/a 1443 n/a n/a n/a BindingDB BindingDB
32 INSR acylated 2-aminobenzimidazole, 14 BD00026820 n/a 145 n/a n/a n/a BindingDB BindingDB
33 INSR CHEMBL1080299 BD50311919 n/a 1493 n/a n/a n/a BindingDB BindingDB
34 INSR CHEMBL1795355 BD50347068 n/a 150 n/a n/a n/a BindingDB BindingDB
35 INSR CHEMBL1796253 BD50347069 n/a 150 n/a n/a n/a BindingDB BindingDB
36 INSR 2-aminobenzimidazole with trans-stilbene, 8x BD00026881 n/a 1500 n/a n/a n/a BindingDB BindingDB
37 INSR CHEMBL1076200 BD50311911 n/a 1506 n/a n/a n/a BindingDB BindingDB
38 INSR CHEMBL1644811 BD50334084 n/a 153 n/a n/a n/a BindingDB BindingDB
39 INSR CHEMBL1087636 BD50311942 n/a 1573 n/a n/a n/a BindingDB BindingDB
40 INSR CHEMBL522328 BD50257856 n/a 160 n/a n/a n/a BindingDB BindingDB
41 INSR CHEMBL1822521 BD50353042 n/a 160 n/a n/a n/a BindingDB BindingDB
42 INSR acylated 2-aminobenzimidazole, 17 BD00026823 n/a 1600 n/a n/a n/a BindingDB BindingDB
43 INSR CHEMBL491686 BD50248413 n/a 1600 n/a n/a n/a BindingDB BindingDB
44 INSR CHEMBL1241670 BD50326007 n/a 1600 n/a n/a n/a BindingDB BindingDB
45 INSR CHEMBL1076474 BD50311936 n/a 1613 n/a n/a n/a BindingDB BindingDB
46 INSR Pyrazine-Pyridine Biheteroaryl 7 BD00006416 n/a 1690 n/a n/a n/a BindingDB BindingDB
47 INSR CHEMBL493319 BD50257697 n/a 1700 n/a n/a n/a BindingDB BindingDB
48 INSR CHEMBL1630118 BD50332493 n/a 1700 n/a n/a n/a BindingDB BindingDB
49 INSR CHEMBL1796242 BD50347055 n/a 1700 n/a n/a n/a BindingDB BindingDB
50 INSR CHEMBL1796241 BD50347054 n/a 180 n/a n/a n/a BindingDB BindingDB
51 INSR CHEMBL485565 BD50274206 n/a 1800 n/a n/a n/a BindingDB BindingDB
52 INSR CHEMBL1076199 BD50311910 n/a 1808 n/a n/a n/a BindingDB BindingDB
53 INSR CHEMBL1076201 BD50311912 n/a 1856 n/a n/a n/a BindingDB BindingDB
54 INSR CHEMBL1642253 BD50334595 n/a 1860 n/a n/a n/a BindingDB BindingDB
55 INSR CHEMBL1822518 BD50353055 n/a 1874 n/a n/a n/a BindingDB BindingDB
56 INSR CHEMBL1642265 BD50334606 n/a 189 n/a n/a n/a BindingDB BindingDB
57 INSR CHEMBL466397 BD50256480 n/a 19 n/a n/a n/a BindingDB BindingDB
58 INSR CHEMBL1822514 BD50353051 n/a 19 n/a n/a n/a BindingDB BindingDB
59 INSR CHEMBL1630108 BD50332491 n/a 1900 n/a n/a n/a BindingDB BindingDB
60 INSR CHEMBL1822512 BD50353050 n/a 194 n/a n/a n/a BindingDB BindingDB
61 INSR 2-aminobenzimidazole with trans-stilbene, 8n BD00026872 n/a 1950 n/a n/a n/a BindingDB BindingDB
62 INSR CHEMBL1088153 BD50311923 n/a 1961 n/a n/a n/a BindingDB BindingDB
63 INSR CHEMBL1079422 BD50311916 n/a 1988 n/a n/a n/a BindingDB BindingDB
64 INSR CHEMBL509032 BD50242742 n/a 20 n/a 1000 n/a BindingDB BindingDB
65 INSR CHEMBL1642132 BD50333558 n/a 20 n/a n/a n/a BindingDB BindingDB
66 INSR CHEMBL1644805 BD50334091 n/a 200 n/a n/a n/a BindingDB BindingDB
67 INSR Pyrrole Analogue 5 BD00015015 n/a 2000 n/a n/a n/a BindingDB BindingDB
68 INSR acylated 2-aminobenzimidazole, 41 BD00026847 n/a 2000 n/a n/a n/a BindingDB BindingDB
69 INSR CHEMBL1822520 BD50353041 n/a 206 n/a n/a n/a BindingDB BindingDB
70 INSR CHEMBL1240829 BD50326003 n/a 2080 n/a n/a n/a BindingDB BindingDB
71 INSR K252a BD00002580 n/a 210 n/a n/a n/a BindingDB BindingDB
72 INSR CHEMBL473761 BD50248351 n/a 2150 n/a n/a n/a BindingDB BindingDB
73 INSR 2-aminobenzimidazole with trans-stilbene, 8s BD00026876 n/a 2200 n/a n/a n/a BindingDB BindingDB
74 INSR CHEMBL520497 BD50267681 n/a 2200 n/a n/a n/a BindingDB BindingDB
75 INSR CHEMBL1240676 BD50326004 n/a 2250 n/a n/a n/a BindingDB BindingDB
76 INSR CHEMBL1076195 BD50311891 n/a 2263 n/a n/a n/a BindingDB BindingDB
77 INSR CHEMBL1644799 BD50334081 n/a 23 n/a n/a n/a BindingDB BindingDB
78 INSR CHEMBL495181 BD50257855 n/a 230 n/a n/a n/a BindingDB BindingDB
79 INSR CHEMBL1642135 BD50333561 n/a 230 n/a n/a n/a BindingDB BindingDB
80 INSR CHEMBL551064 BD50296348 n/a 2300 n/a n/a n/a BindingDB BindingDB
81 INSR CHEMBL1642145 BD50333571 n/a 2300 n/a n/a n/a BindingDB BindingDB
82 INSR CHEMBL1644815 BD50334087 n/a 231 n/a n/a n/a BindingDB BindingDB
83 INSR CHEMBL1642264 BD50334605 n/a 233 n/a n/a n/a BindingDB BindingDB
84 INSR CHEMBL447107 BD50263515 n/a 2345 n/a n/a n/a BindingDB BindingDB
85 INSR CHEMBL519698 BD50274249 n/a 235 n/a n/a n/a BindingDB BindingDB
86 INSR CHEMBL1760057 BD50340143 n/a 24 n/a n/a n/a BindingDB BindingDB
87 INSR acylated 2-aminobenzimidazole, 15 BD00026821 n/a 240 n/a n/a n/a BindingDB BindingDB
88 INSR acylated 2-aminobenzimidazole, 38 BD00026844 n/a 2400 n/a n/a n/a BindingDB BindingDB
89 INSR 1-Acyl-1H-[1,2,4]triazole-3,5-diamine Analogue 3f BD00006870 n/a 2400 n/a n/a n/a BindingDB BindingDB
90 INSR CHEMBL458997 BD50334594 n/a 25 n/a n/a n/a BindingDB BindingDB
91 INSR CHEMBL1630112 BD50332485 n/a 2500 n/a n/a n/a BindingDB BindingDB
92 INSR CHEMBL1688360 BD50339061 n/a 260 n/a n/a n/a BindingDB BindingDB
93 INSR Anilinoquinazoline deriv. 9 BD00004626 n/a 2600 n/a n/a n/a BindingDB BindingDB
94 INSR CHEMBL489083 BD50246774 n/a 2600 n/a n/a n/a BindingDB BindingDB
95 INSR CHEMBL1076194 BD50311890 n/a 2628 n/a n/a n/a BindingDB BindingDB
96 INSR CHEMBL1822523 BD50353044 n/a 266 n/a n/a n/a BindingDB BindingDB
97 INSR CHEMBL1642255 BD50334597 n/a 2694 n/a n/a n/a BindingDB BindingDB
98 INSR CHEMBL474543 BD50248230 n/a 2700 n/a n/a n/a BindingDB BindingDB
99 INSR CHEMBL370800 BD50181669 5300 27000 n/a n/a n/a BindingDB BindingDB
100 INSR CHEMBL1076465 BD50311943 n/a 2768 n/a n/a n/a BindingDB BindingDB
101 INSR CHEMBL558708 BD50296347 n/a 2800 n/a n/a n/a BindingDB BindingDB
102 INSR CHEMBL1630114 BD50332487 n/a 2800 n/a n/a n/a BindingDB BindingDB
103 INSR CHEMBL1087127 BD50311897 n/a 29 n/a n/a n/a BindingDB BindingDB
104 INSR CHEMBL1822511 BD50353049 n/a 295 n/a n/a n/a BindingDB BindingDB
105 INSR CHEMBL1760035 BD50340121 n/a 3 n/a n/a n/a BindingDB BindingDB
106 INSR CHEMBL1644804 BD50334088 n/a 30 n/a n/a n/a BindingDB BindingDB
107 INSR CHEMBL1642142 BD50333568 n/a 300 n/a n/a n/a BindingDB BindingDB
108 INSR CHEMBL1738841 BD50340484 n/a 300 n/a n/a n/a BindingDB BindingDB
109 INSR CHEMBL1288160 BD50332091 n/a 3000 n/a n/a n/a BindingDB BindingDB
110 INSR CHEMBL1630115 BD50332488 n/a 3000 n/a n/a n/a BindingDB BindingDB
111 INSR CHEMBL1076470 BD50311932 n/a 3012 n/a n/a n/a BindingDB BindingDB
112 INSR CHEMBL521695 BD50257803 n/a 310 n/a n/a n/a BindingDB BindingDB
113 INSR CHEMBL1779202 BD50344664 n/a 310 n/a n/a n/a BindingDB BindingDB
114 INSR CHEMBL1076469 BD50311931 n/a 3109 n/a n/a n/a BindingDB BindingDB
115 INSR CHEMBL1076478 BD50311893 n/a 3162 n/a n/a n/a BindingDB BindingDB
116 INSR CHEMBL1076197 BD50311908 n/a 3194 n/a n/a n/a BindingDB BindingDB
117 INSR CHEMBL494027 BD50257917 n/a 320 n/a n/a n/a BindingDB BindingDB
118 INSR CHEMBL522682 BD50257918 n/a 320 n/a n/a n/a BindingDB BindingDB
119 INSR CHEMBL460389 BD50274000 n/a 320 n/a n/a n/a BindingDB BindingDB
120 INSR CHEMBL1688362 BD50339063 n/a 320 n/a n/a n/a BindingDB BindingDB
121 INSR 2-aminobenzimidazole with trans-stilbene, 8c BD00026860 n/a 3250 n/a n/a n/a BindingDB BindingDB
122 INSR CHEMBL1822516 BD50353053 n/a 326 n/a n/a n/a BindingDB BindingDB
123 INSR 2-aminobenzimidazole with trans-stilbene, 8v BD00026879 n/a 330 n/a n/a n/a BindingDB BindingDB
124 INSR 2-aminobenzimidazole with trans-stilbene, 8q BD00026874 n/a 3300 n/a n/a n/a BindingDB BindingDB
125 INSR CHEMBL1088429 BD50311928 n/a 3332 n/a n/a n/a BindingDB BindingDB
126 INSR CHEMBL1644808 BD50334092 n/a 334 n/a n/a n/a BindingDB BindingDB
127 INSR CHEMBL1834657 BD50355393 n/a 3371 n/a n/a n/a BindingDB BindingDB
128 INSR CHEMBL1644801 BD50334090 n/a 34 n/a n/a n/a BindingDB BindingDB
129 INSR CHEMBL1076196 BD50311892 n/a 3486 n/a n/a n/a BindingDB BindingDB
130 INSR CHEMBL1822513 BD50353056 n/a 35 n/a n/a n/a BindingDB BindingDB
131 INSR CHEMBL493106 BD50257655 n/a 350 n/a n/a n/a BindingDB BindingDB
132 INSR CHEMBL551570 BD50294542 n/a 3500 n/a n/a n/a BindingDB BindingDB
133 INSR CHEMBL1642263 BD50334604 n/a 351 n/a n/a n/a BindingDB BindingDB
134 INSR CHEMBL1822522 BD50353043 n/a 357 n/a n/a n/a BindingDB BindingDB
135 INSR CHEMBL522871 BD50257805 n/a 360 n/a n/a n/a BindingDB BindingDB
136 INSR CHEMBL199723 BD50181672 >20000 3600 n/a n/a n/a BindingDB BindingDB
137 INSR 2-aminobenzimidazole with trans-stilbene, 9e BD00026884 n/a 3600 n/a n/a n/a BindingDB BindingDB
138 INSR CHEMBL1630109 BD50332494 n/a 3600 n/a n/a n/a BindingDB BindingDB
139 INSR CHEMBL1821735 BD50353039 n/a 366 n/a n/a n/a BindingDB BindingDB
140 INSR CHEMBL1644809 BD50334089 n/a 369 n/a n/a n/a BindingDB BindingDB
141 INSR CHEMBL1642141 BD50333567 n/a 370 n/a n/a n/a BindingDB BindingDB
142 INSR Pyrido[2,3-d]pyrimidin-5-one, 37 BD00027909 n/a 3700 n/a n/a n/a BindingDB BindingDB
143 INSR CHEMBL1630110 BD50332492 n/a 3700 n/a n/a n/a BindingDB BindingDB
144 INSR CHEMBL1076466 BD50311944 n/a 3760 n/a n/a n/a BindingDB BindingDB
145 INSR acylated 2-aminobenzimidazole, 22 BD00026828 n/a 380 n/a n/a n/a BindingDB BindingDB
146 INSR CHEMBL1241669 BD50326005 n/a 380 n/a n/a n/a BindingDB BindingDB
147 INSR acylated 2-aminobenzimidazole, 24 BD00026830 n/a 3800 n/a n/a n/a BindingDB BindingDB
148 INSR 2-aminobenzimidazole with trans-stilbene, 8w BD00026880 n/a 3800 n/a n/a n/a BindingDB BindingDB
149 INSR CHEMBL492990 BD50257858 n/a 390 n/a n/a n/a BindingDB BindingDB
150 INSR CHEMBL483403 BD50274340 n/a 3900 n/a n/a n/a BindingDB BindingDB
151 INSR CHEMBL1822519 BD50353040 n/a 391 n/a n/a n/a BindingDB BindingDB
152 INSR CHEMBL1086731 BD50311921 n/a 4 n/a n/a n/a BindingDB BindingDB
153 INSR CHEMBL1644798 BD50334080 n/a 4 n/a n/a n/a BindingDB BindingDB
154 INSR CHEMBL493928 BD50257699 n/a 400 n/a n/a n/a BindingDB BindingDB
155 INSR CHEMBL522711 BD50257857 n/a 400 n/a n/a n/a BindingDB BindingDB
156 INSR 2-aminobenzimidazole with trans-stilbene, 8g BD00026863 n/a 4000 n/a n/a n/a BindingDB BindingDB
157 INSR CHEMBL176078 BD50162978 n/a 4000 n/a n/a n/a BindingDB BindingDB
158 INSR CHEMBL1644813 BD50334096 n/a 404 n/a n/a n/a BindingDB BindingDB
159 INSR CHEMBL1076436 BD50311926 n/a 409 n/a n/a n/a BindingDB BindingDB
160 INSR CHEMBL1076471 BD50311933 n/a 4156 n/a n/a n/a BindingDB BindingDB
161 INSR CHEMBL177298 BD50162973 n/a 420 n/a n/a n/a BindingDB BindingDB
162 INSR CHEMBL494743 BD50257962 n/a 420 n/a n/a n/a BindingDB BindingDB
163 INSR CHEMBL1796258 BD50347071 n/a 430 n/a n/a n/a BindingDB BindingDB
164 INSR 2-aminobenzimidazole with trans-stilbene, 8r BD00026875 n/a 4300 n/a n/a n/a BindingDB BindingDB
165 INSR CHEMBL1087638 BD50311894 n/a 4401 n/a n/a n/a BindingDB BindingDB
166 INSR 2-aminobenzimidazole with trans-stilbene, 9d BD00026883 n/a 4500 n/a n/a n/a BindingDB BindingDB
167 INSR CHEMBL1796257 BD50347070 n/a 460 n/a n/a n/a BindingDB BindingDB
168 INSR CHEMBL1823221 BD50352760 n/a 460 n/a n/a n/a BindingDB BindingDB
169 INSR CHEMBL1688361 BD50339062 n/a 48 n/a n/a n/a BindingDB BindingDB
170 INSR 2-aminobenzimidazole with trans-stilbene, 8b BD00026859 n/a 480 n/a n/a n/a BindingDB BindingDB
171 INSR CHEMBL522849 BD50257698 n/a 480 n/a n/a n/a BindingDB BindingDB
172 INSR CHEMBL493537 BD50257755 n/a 480 n/a n/a n/a BindingDB BindingDB
173 INSR CHEMBL436509 BD50181670 8800 4800 n/a n/a n/a BindingDB BindingDB
174 INSR CHEMBL1642148 BD50333574 n/a 490 n/a n/a n/a BindingDB BindingDB
175 INSR 2-aminobenzimidazole with trans-stilbene, 8p BD00026873 n/a 4900 n/a n/a n/a BindingDB BindingDB
176 INSR CHEMBL485402 BD50274248 n/a 4900 n/a n/a n/a BindingDB BindingDB
177 INSR CHEMBL507714 BD50256478 n/a 5 n/a n/a n/a BindingDB BindingDB
178 INSR CHEMBL494135 BD50257753 n/a 500 n/a n/a n/a BindingDB BindingDB
179 INSR CHEMBL1642144 BD50333570 n/a 500 n/a n/a n/a BindingDB BindingDB
180 INSR Purvalanol A BD00027216 n/a 5000 n/a n/a n/a BindingDB BindingDB
181 INSR CHEMBL1164453 BD50320978 n/a 5010 n/a n/a n/a BindingDB BindingDB
182 INSR CHEMBL1642259 BD50334600 n/a 504 n/a n/a n/a BindingDB BindingDB
183 INSR acylated 2-aminobenzimidazole, 25 BD00026831 n/a 51 n/a n/a n/a BindingDB BindingDB
184 INSR CHEMBL564417 BD50296350 n/a 51 n/a n/a n/a BindingDB BindingDB
185 INSR CHEMBL447317 BD50246732 n/a 5100 n/a n/a n/a BindingDB BindingDB
186 INSR CHEMBL1240677 BD50326006 n/a 5150 n/a n/a n/a BindingDB BindingDB
187 INSR CHEMBL473250 BD50263514 n/a 5165 n/a n/a n/a BindingDB BindingDB
188 INSR acylated 2-aminobenzimidazole, 37 BD00026843 n/a 5200 n/a n/a n/a BindingDB BindingDB
189 INSR CHEMBL1796245 BD50347058 n/a 540 n/a n/a n/a BindingDB BindingDB
190 INSR Pyrrole Analogue 2 BD00015012 n/a 5400 n/a n/a n/a BindingDB BindingDB
191 INSR CHEMBL1081090 BD50311903 n/a 5435 n/a n/a n/a BindingDB BindingDB
192 INSR CHEMBL175862 BD50162976 n/a 550 n/a n/a n/a BindingDB BindingDB
193 INSR CHEMBL493007 BD50257915 n/a 550 n/a n/a n/a BindingDB BindingDB
194 INSR CHEMBL485233 BD50274247 n/a 550 n/a n/a n/a BindingDB BindingDB
195 INSR CHEMBL520312 BD50274341 n/a 550 n/a n/a n/a BindingDB BindingDB
196 INSR CHEMBL483602 BD50274394 n/a 550 n/a n/a n/a BindingDB BindingDB
197 INSR CHEMBL1642136 BD50333562 n/a 550 n/a n/a n/a BindingDB BindingDB
198 INSR CHEMBL493318 BD50257696 n/a 5500 n/a n/a n/a BindingDB BindingDB
199 INSR CHEMBL1630113 BD50332486 n/a 5500 n/a n/a n/a BindingDB BindingDB
200 INSR acylated 2-aminobenzimidazole, 1 BD00026811 n/a 560 n/a n/a n/a BindingDB BindingDB
201 INSR CHEMBL1642143 BD50333569 n/a 560 n/a n/a n/a BindingDB BindingDB
202 INSR acylated 2-aminobenzimidazole, 6 BD00026812 n/a 5600 n/a n/a n/a BindingDB BindingDB
203 INSR CHEMBL1088028 BD50311900 n/a 5629 n/a n/a n/a BindingDB BindingDB
204 INSR CHEMBL494136 BD50257754 n/a 570 n/a n/a n/a BindingDB BindingDB
205 INSR CHEMBL1081436 BD50311905 n/a 5708 n/a n/a n/a BindingDB BindingDB
206 INSR CHEMBL1642261 BD50334602 n/a 573 n/a n/a n/a BindingDB BindingDB
207 INSR CHEMBL1164264 BD50320970 n/a 5750 n/a n/a n/a BindingDB BindingDB
208 INSR acylated 2-aminobenzimidazole, 12 BD00026818 n/a 5800 n/a n/a n/a BindingDB BindingDB
209 INSR CHEMBL1076437 BD50311927 n/a 588 n/a n/a n/a BindingDB BindingDB
210 INSR CHEMBL1076533 BD50311904 n/a 5935 n/a n/a n/a BindingDB BindingDB
211 INSR CHEMBL495026 BD50257804 n/a 600 n/a n/a n/a BindingDB BindingDB
212 INSR CHEMBL551264 BD50296357 n/a 610 n/a n/a n/a BindingDB BindingDB
213 INSR acylated 2-aminobenzimidazole, 16 BD00026822 n/a 6100 n/a n/a n/a BindingDB BindingDB
214 INSR CHEMBL1642260 BD50334601 n/a 62 n/a n/a n/a BindingDB BindingDB
215 INSR CHEMBL1076433 BD50311924 n/a 63 n/a n/a n/a BindingDB BindingDB
216 INSR acylated 2-aminobenzimidazole, 23 BD00026829 n/a 630 n/a n/a n/a BindingDB BindingDB
217 INSR CHEMBL514941 BD50248350 n/a 630 n/a n/a n/a BindingDB BindingDB
218 INSR CHEMBL488271 BD50246776 n/a 6300 n/a n/a n/a BindingDB BindingDB
219 INSR CHEMBL1796243 BD50347056 n/a 6300 n/a n/a n/a BindingDB BindingDB
220 INSR CHEMBL1079945 BD50311917 n/a 661 n/a n/a n/a BindingDB BindingDB
221 INSR CHEMBL1688363 BD50339064 n/a 68 n/a n/a n/a BindingDB BindingDB
222 INSR CHEMBL518803 BD50248148 n/a 6950 n/a n/a n/a BindingDB BindingDB
223 INSR CHEMBL448929 BD50256479 n/a 7 n/a n/a n/a BindingDB BindingDB
224 INSR CHEMBL493107 BD50257656 n/a 700 n/a n/a n/a BindingDB BindingDB
225 INSR CHEMBL1688359 BD50339060 n/a 700 n/a n/a n/a BindingDB BindingDB
226 INSR CHEMBL202830 BD50181682 n/a 7000 n/a n/a n/a BindingDB BindingDB
227 INSR CHEMBL1258913 BD50327912 n/a 7012 n/a n/a n/a BindingDB BindingDB
228 INSR CHEMBL1164177 BD50320967 n/a 7080 n/a n/a n/a BindingDB BindingDB
229 INSR CHEMBL1796247 BD50347062 n/a 710 n/a n/a n/a BindingDB BindingDB
230 INSR CHEMBL1630116 BD50332489 n/a 7100 n/a n/a n/a BindingDB BindingDB
231 INSR CHEMBL1087002 BD50311896 n/a 7121 n/a n/a n/a BindingDB BindingDB
232 INSR BMS-536924 BD00027879 n/a 73 n/a n/a n/a BindingDB BindingDB
233 INSR CHEMBL562724 BD50296349 n/a 73 n/a n/a n/a BindingDB BindingDB
234 INSR CHEMBL1644812 BD50334085 n/a 730 n/a n/a n/a BindingDB BindingDB
235 INSR CHEMBL1630107 BD50332483 n/a 7340 n/a n/a n/a BindingDB BindingDB
236 INSR CHEMBL1796246 BD50347061 n/a 740 n/a n/a n/a BindingDB BindingDB
237 INSR CHEMBL1076432 BD50311920 n/a 746 n/a n/a n/a BindingDB BindingDB
238 INSR CHEMBL1086860 BD50311922 n/a 75 n/a n/a n/a BindingDB BindingDB
239 INSR CHEMBL1667935 BD50336317 n/a 76 n/a n/a n/a BindingDB BindingDB
240 INSR CHEMBL1076193 BD50311889 n/a 7631 n/a n/a n/a BindingDB BindingDB
241 INSR CHEMBL1796256 BD50347060 n/a 77 n/a n/a n/a BindingDB BindingDB
242 INSR CHEMBL491677 BD50248464 n/a 7900 n/a n/a n/a BindingDB BindingDB
243 INSR CHEMBL1644802 BD50334082 n/a 8 n/a n/a n/a BindingDB BindingDB
244 INSR CHEMBL162 BD50059889 n/a 8.5 73 n/a n/a BindingDB BindingDB
245 INSR CHEMBL1090360 BD50315888 n/a 80 n/a n/a n/a BindingDB BindingDB
246 INSR CHEMBL1642139 BD50333565 n/a 800 n/a n/a n/a BindingDB BindingDB
247 INSR CHEMBL1822527 BD50353048 n/a 809 n/a n/a n/a BindingDB BindingDB
248 INSR CHEMBL1075628 BD50311925 n/a 818 n/a n/a n/a BindingDB BindingDB
249 INSR CHEMBL1642138 BD50333564 n/a 820 n/a n/a n/a BindingDB BindingDB
250 INSR CHEMBL1644814 BD50334093 n/a 840 n/a n/a n/a BindingDB BindingDB
251 INSR CHEMBL1796251 BD50347066 n/a 840 n/a n/a n/a BindingDB BindingDB
252 INSR CHEMBL485232 BD50274246 n/a 850 n/a n/a n/a BindingDB BindingDB
253 INSR CHEMBL1809044 BD50349687 n/a 9 n/a n/a n/a BindingDB BindingDB
254 INSR CHEMBL460746 BD50248085 n/a 900 n/a n/a n/a BindingDB BindingDB
255 INSR CHEMBL604159 BD50308355 n/a 905 n/a n/a n/a BindingDB BindingDB
256 INSR CHEMBL1796244 BD50347057 n/a 920 n/a n/a n/a BindingDB BindingDB
257 INSR CHEMBL494993 BD50257806 n/a 93 n/a n/a n/a BindingDB BindingDB
258 INSR CHEMBL1642146 BD50333572 n/a 930 n/a n/a n/a BindingDB BindingDB
259 INSR CHEMBL1796249 BD50347064 n/a 930 n/a n/a n/a BindingDB BindingDB
260 INSR Pyrido[2,3-d]pyrimidin-5-one, 36 BD00027908 n/a 9300 n/a n/a n/a BindingDB BindingDB
261 INSR CHEMBL1164262 BD50320968 n/a 9330 n/a n/a n/a BindingDB BindingDB
262 INSR CHEMBL1822524 BD50353045 n/a 934 n/a n/a n/a BindingDB BindingDB
263 INSR CHEMBL522785 BD50248414 n/a 940 n/a n/a n/a BindingDB BindingDB
264 INSR CHEMBL492931 BD50257549 n/a 940 n/a n/a n/a BindingDB BindingDB
265 INSR CHEMBL483397 BD50274338 n/a 95 n/a n/a n/a BindingDB BindingDB
266 INSR CHEMBL199886 BD50174686 n/a 9500 n/a n/a n/a BindingDB BindingDB
267 INSR 2-aminobenzimidazole with trans-stilbene, 8f BD00026862 n/a 970 n/a n/a n/a BindingDB BindingDB
268 INSR CHEMBL512933 BD50248117 n/a 9700 n/a n/a n/a BindingDB BindingDB
269 INSR 1-Acyl-1H-[1,2,4]triazole-3,5-diamine Analogue 3c BD00006867 n/a 9800 n/a n/a n/a BindingDB BindingDB
270 INSR CHEMBL1241764 BD50326008 n/a 9900 n/a n/a n/a BindingDB BindingDB
271 INSR CHEBI:305251 BD50117315 n/a <0.3 n/a n/a n/a BindingDB BindingDB
272 INSR GSK_1838705A GSK_1838705A n/a n/a 1.7 n/a n/a NB2011DRx NB2011DRx
273 INSR Staurosporine Staurosporine n/a n/a 110 n/a n/a NB2008 NB2008
274 INSR Staurosporine Staurosporine n/a n/a 110 n/a n/a NB2011DRx NB2011DRx
275 INSR CHEMBL603469 BD50308060 n/a n/a 1100 n/a n/a BindingDB BindingDB
276 INSR CEP_701 CEP_701 n/a n/a 1100 n/a n/a NB2011DRx NB2011DRx
277 INSR R406 R406 n/a n/a 1100 n/a n/a NB2011DRx NB2011DRx
278 INSR cid_10138259 BD00031095 n/a n/a 1200 n/a n/a BindingDB BindingDB
279 INSR SU_14813 SU_14813 n/a n/a 1200 n/a n/a NB2008 NB2008
280 INSR SU_14813 SU_14813 n/a n/a 1200 n/a n/a NB2011DRx NB2011DRx
281 INSR SU11248 BD00004814 n/a n/a 180 n/a n/a BindingDB BindingDB
282 INSR TAE_684 TAE_684 n/a n/a 2.4 n/a n/a NB2011DRx NB2011DRx
283 INSR EXEL_2880 EXEL_2880 n/a n/a 210 n/a n/a NB2011DRx NB2011DRx
284 INSR AST_487 AST_487 n/a n/a 2200 n/a n/a NB2011DRx NB2011DRx
285 INSR PHA_665752 PHA_665752 n/a n/a 2300 n/a n/a NB2011DRx NB2011DRx
286 INSR BIBF_1120der BIBF_1120der n/a n/a 24 n/a n/a NB2011DRx NB2011DRx
287 INSR HKI_272 HKI_272 n/a n/a 3000 n/a n/a NB2011DRx NB2011DRx
288 INSR JNJ_28312141 JNJ_28312141 n/a n/a 330 n/a n/a NB2011DRx NB2011DRx
289 INSR Crizotinib Crizotinib n/a n/a 340 n/a n/a NB2011DRx NB2011DRx
290 INSR KW_2449 KW_2449 n/a n/a 400 n/a n/a NB2011DRx NB2011DRx
291 INSR Sunitinib Sunitinib n/a n/a 500 n/a n/a NB2008 NB2008
292 INSR Sunitinib Sunitinib n/a n/a 500 n/a n/a NB2011DRx NB2011DRx
293 INSR VX-680 BD00013534 n/a n/a 506 n/a n/a BindingDB BindingDB
294 INSR VX_680 VX_680 n/a n/a 630 n/a n/a NB2008 NB2008
295 INSR VX_680 VX_680 n/a n/a 630 n/a n/a NB2011DRx NB2011DRx
296 INSR Staurosporine BD00002579 n/a n/a 73 n/a n/a BindingDB BindingDB
297 INSR TG_101348 TG_101348 n/a n/a 850 n/a n/a NB2011DRx NB2011DRx
298 INSR Myricetin BD00015236 2600 n/a n/a n/a n/a BindingDB BindingDB
299 INSR 351 351 n/a n/a n/a n/a n/a PDB PDB
300 INSR CHEMBL117206 BD50092143 n/a n/a n/a 300 n/a BindingDB BindingDB
301 INSR CHEMBL331137 BD50092144 n/a n/a n/a 7000 n/a BindingDB BindingDB
302 INSR CHEMBL116907 BD50092146 n/a n/a n/a 1500 n/a BindingDB BindingDB
303 INSR CHEMBL432971 BD50092147 n/a n/a n/a 6000 n/a BindingDB BindingDB
304 INSR CHEMBL117440 BD50092148 n/a n/a n/a 1000 n/a BindingDB BindingDB
305 INSR CHEMBL18879 BD50092149 n/a n/a n/a 5000 n/a BindingDB BindingDB
306 INSR CHEMBL116306 BD50092150 n/a n/a n/a 300 n/a BindingDB BindingDB
307 INSR ACP ACP n/a n/a n/a n/a n/a PDB PDB
308 INSR ANP ANP n/a n/a n/a n/a n/a PDB PDB
309 INSR ATP ATP n/a n/a n/a n/a n/a PDB PDB
310 INSR CAS135897_06_2 CAS135897_06_2 n/a n/a n/a n/a 17.19 NB2011RBC NB2011RBC
311 INSR CAS244148_46_7 CAS244148_46_7 n/a n/a n/a n/a 17.85 NB2011RBC NB2011RBC
312 INSR CAS326914_10_7 CAS326914_10_7 n/a n/a n/a n/a 30.12 NB2011RBC NB2011RBC
313 INSR CAS331253_86_2 CAS331253_86_2 n/a n/a n/a n/a 32.26 NB2011RBC NB2011RBC
314 INSR CAS404828_08_6 CAS404828_08_6 n/a n/a n/a n/a 31.56 NB2011RBC NB2011RBC
315 INSR CAS62996_74_1 CAS62996_74_1 n/a n/a n/a n/a 3.14 NB2011RBC NB2011RBC
316 INSR CAS639089_54_6 CAS639089_54_6 n/a n/a n/a n/a 43.5 NB2011RBC NB2011RBC
317 INSR CAS854171_35_0 CAS854171_35_0 n/a n/a n/a n/a 44.92 NB2011RBC NB2011RBC
318 INSR CAS97161_97_2 CAS97161_97_2 n/a n/a n/a n/a 32.16 NB2011RBC NB2011RBC
319 INSR GS2 GS2 n/a n/a n/a n/a n/a PDB PDB
320 INSR GS3 GS3 n/a n/a n/a n/a n/a PDB PDB
321 INSR S91 S91 n/a n/a n/a n/a n/a PDB PDB