Summary of query kinase
Query kinase MAP2K1 (Q02750)
Kinase group STE
Number of inhibitors 353
Index Target Inhibitor Inhibitor 2D Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) POC Source Link
0 MAP2K1 CHEMBL106489 BD50132262 n/a 1 n/a n/a n/a BindingDB BindingDB
1 MAP2K1 3-cyanoquinoline, 9 BD00028124 n/a 1.1 n/a n/a n/a BindingDB BindingDB
2 MAP2K1 CHEMBL337728 BD50109282 n/a 10 n/a n/a n/a BindingDB BindingDB
3 MAP2K1 CHEMBL321045 BD50132265 n/a 10 n/a n/a n/a BindingDB BindingDB
4 MAP2K1 CHEMBL485238 BD50274335 n/a 10 n/a n/a n/a BindingDB BindingDB
5 MAP2K1 CHEMBL80837 BD50145191 n/a 10000 n/a n/a n/a BindingDB BindingDB
6 MAP2K1 CHEMBL426840 BD50180567 n/a 105 n/a n/a n/a BindingDB BindingDB
7 MAP2K1 CHEMBL384784 BD50194027 n/a 107 n/a 37 n/a BindingDB BindingDB
8 MAP2K1 CHEMBL485237 BD50274333 n/a 11 n/a n/a n/a BindingDB BindingDB
9 MAP2K1 CHEMBL1170802 BD50321561 n/a 11 n/a n/a n/a BindingDB BindingDB
10 MAP2K1 CHEMBL1170805 BD50321567 n/a 11 n/a n/a n/a BindingDB BindingDB
11 MAP2K1 CHEMBL31149 BD50099975 n/a 110 n/a n/a n/a BindingDB BindingDB
12 MAP2K1 CHEMBL318939 BD50072150 n/a 1100 n/a n/a n/a BindingDB BindingDB
13 MAP2K1 CHEMBL285956 BD50099986 n/a 1100 n/a n/a n/a BindingDB BindingDB
14 MAP2K1 CHEMBL202545 BD50176597 n/a 1110 n/a n/a n/a BindingDB BindingDB
15 MAP2K1 CHEMBL201691 BD50180568 n/a 118 n/a n/a n/a BindingDB BindingDB
16 MAP2K1 CHEMBL489058 BD50274385 n/a 12 n/a n/a n/a BindingDB BindingDB
17 MAP2K1 CHEMBL217833 BD50194038 n/a 120 n/a 95 n/a BindingDB BindingDB
18 MAP2K1 CHEMBL217130 BD50194047 n/a 120 n/a 100 n/a BindingDB BindingDB
19 MAP2K1 CHEMBL377591 BD50187823 n/a 1230 n/a n/a n/a BindingDB BindingDB
20 MAP2K1 CHEMBL201379 BD50180574 n/a 124 n/a n/a n/a BindingDB BindingDB
21 MAP2K1 CHEMBL98131 BD50095234 n/a 125 n/a n/a n/a BindingDB BindingDB
22 MAP2K1 CHEMBL1171013 BD50321572 n/a 13 n/a n/a n/a BindingDB BindingDB
23 MAP2K1 CHEMBL1169631 BD50321577 n/a 13 n/a n/a n/a BindingDB BindingDB
24 MAP2K1 CHEMBL214977 BD50194042 n/a 137 n/a 118 n/a BindingDB BindingDB
25 MAP2K1 CHEMBL209489 BD50187805 n/a 1390 n/a n/a n/a BindingDB BindingDB
26 MAP2K1 CHEMBL30790 BD50099984 n/a 14 n/a n/a n/a BindingDB BindingDB
27 MAP2K1 CHEMBL202286 BD50176588 n/a 14 n/a n/a n/a BindingDB BindingDB
28 MAP2K1 CHEMBL371693 BD50180572 n/a 14 n/a n/a n/a BindingDB BindingDB
29 MAP2K1 CHEMBL425980 BD50194067 n/a 140 n/a 30 n/a BindingDB BindingDB
30 MAP2K1 CHEMBL97724 BD50072144 n/a 1400 n/a n/a n/a BindingDB BindingDB
31 MAP2K1 CHEMBL375410 BD50187820 n/a 1440 n/a n/a n/a BindingDB BindingDB
32 MAP2K1 CHEMBL213562 BD50187862 n/a 1440 n/a n/a n/a BindingDB BindingDB
33 MAP2K1 CHEMBL385203 BD50194029 n/a 145 n/a 200 n/a BindingDB BindingDB
34 MAP2K1 CHEMBL209520 BD50187860 n/a 1450 n/a n/a n/a BindingDB BindingDB
35 MAP2K1 CHEMBL200969 BD50176575 n/a 147 n/a n/a n/a BindingDB BindingDB
36 MAP2K1 CHEMBL214636 BD50194060 n/a 147 n/a 284 n/a BindingDB BindingDB
37 MAP2K1 CHEMBL203258 BD50180561 n/a 15 n/a n/a n/a BindingDB BindingDB
38 MAP2K1 CHEMBL217117 BD50194044 n/a 150 n/a 278 n/a BindingDB BindingDB
39 MAP2K1 CHEMBL491434 BD50264738 n/a 1500 n/a n/a n/a BindingDB BindingDB
40 MAP2K1 CHEMBL491635 BD50264741 n/a 1500 n/a n/a n/a BindingDB BindingDB
41 MAP2K1 CHEMBL1684068 BD50337927 n/a 16 n/a n/a n/a BindingDB BindingDB
42 MAP2K1 CHEMBL31639 BD50099977 n/a 160 n/a n/a n/a BindingDB BindingDB
43 MAP2K1 CHEMBL413636 BD50194049 n/a 160 n/a 130 n/a BindingDB BindingDB
44 MAP2K1 CHEMBL382616 BD50176584 n/a 168 n/a n/a n/a BindingDB BindingDB
45 MAP2K1 CHEMBL281662 BD50099979 n/a 18 n/a n/a n/a BindingDB BindingDB
46 MAP2K1 CHEMBL383108 BD50176580 n/a 18 n/a n/a n/a BindingDB BindingDB
47 MAP2K1 CHEMBL199860 BD50180562 n/a 18 n/a n/a n/a BindingDB BindingDB
48 MAP2K1 CHEMBL1169814 BD50321564 n/a 18 n/a n/a n/a BindingDB BindingDB
49 MAP2K1 CHEMBL1169999 BD50321570 n/a 18 n/a n/a n/a BindingDB BindingDB
50 MAP2K1 CHEMBL1684800 BD50338873 n/a 18.19 n/a n/a n/a BindingDB BindingDB
51 MAP2K1 CHEMBL490423 BD50264742 n/a 1800 n/a n/a n/a BindingDB BindingDB
52 MAP2K1 CHEMBL201251 BD50176601 n/a 181 n/a n/a n/a BindingDB BindingDB
53 MAP2K1 BMS-536924 BD00027879 n/a 182 n/a n/a n/a BindingDB BindingDB
54 MAP2K1 CHEMBL97463 BD50095230 n/a 185 n/a n/a n/a BindingDB BindingDB
55 MAP2K1 CHEMBL520142 BD50274384 n/a 19 n/a n/a n/a BindingDB BindingDB
56 MAP2K1 CHEMBL1171012 BD50321568 n/a 19 n/a n/a n/a BindingDB BindingDB
57 MAP2K1 CHEMBL1171015 BD50321574 n/a 19 n/a n/a n/a BindingDB BindingDB
58 MAP2K1 CHEMBL30540 BD50099974 n/a 190 n/a n/a n/a BindingDB BindingDB
59 MAP2K1 CHEMBL203096 BD50176583 n/a 190 n/a n/a n/a BindingDB BindingDB
60 MAP2K1 CHEMBL316635 BD50072146 n/a 1900 n/a n/a n/a BindingDB BindingDB
61 MAP2K1 CHEMBL94565 BD50072157 n/a 1900 n/a n/a n/a BindingDB BindingDB
62 MAP2K1 CHEMBL522129 BD50264739 n/a 1900 n/a n/a n/a BindingDB BindingDB
63 MAP2K1 CHEMBL382456 BD50176591 n/a 191 n/a n/a n/a BindingDB BindingDB
64 MAP2K1 3-cyanoquinoline, 8 BD00028123 n/a 2 n/a n/a n/a BindingDB BindingDB
65 MAP2K1 CHEMBL105442 BD50132260 n/a 2 n/a n/a n/a BindingDB BindingDB
66 MAP2K1 CHEMBL105642 BD50132261 n/a 2 n/a n/a n/a BindingDB BindingDB
67 MAP2K1 CHEMBL102374 BD50132264 n/a 2 n/a n/a n/a BindingDB BindingDB
68 MAP2K1 CHEMBL105220 BD50132266 n/a 2 n/a n/a n/a BindingDB BindingDB
69 MAP2K1 CHEMBL1668411 BD50336457 n/a 2 n/a n/a n/a BindingDB BindingDB
70 MAP2K1 CHEMBL414139 BD50095232 n/a 2.4 n/a n/a n/a BindingDB BindingDB
71 MAP2K1 CHEMBL162 BD50059889 n/a 2.5 21 n/a n/a BindingDB BindingDB
72 MAP2K1 CHEMBL30728 BD50099987 n/a 2.7 n/a n/a n/a BindingDB BindingDB
73 MAP2K1 CHEMBL31143 BD50099978 n/a 20 n/a n/a n/a BindingDB BindingDB
74 MAP2K1 CHEMBL214734 BD50194048 n/a 20 n/a 1450 n/a BindingDB BindingDB
75 MAP2K1 CHEMBL214613 BD50194053 n/a 20 n/a 42 n/a BindingDB BindingDB
76 MAP2K1 CHEMBL521502 BD50274334 n/a 20 n/a n/a n/a BindingDB BindingDB
77 MAP2K1 CHEMBL1169813 BD50321562 n/a 20 n/a n/a n/a BindingDB BindingDB
78 MAP2K1 CHEMBL1170804 BD50321566 n/a 20 n/a n/a n/a BindingDB BindingDB
79 MAP2K1 CHEMBL282976 BD50099992 n/a 200 n/a n/a n/a BindingDB BindingDB
80 MAP2K1 CHEMBL216500 BD50194043 n/a 200 n/a 6190 n/a BindingDB BindingDB
81 MAP2K1 CHEMBL495729 BD50265035 n/a 200 n/a n/a n/a BindingDB BindingDB
82 MAP2K1 CHEMBL95400 BD50072161 n/a 2000 n/a n/a n/a BindingDB BindingDB
83 MAP2K1 CHEMBL35482 BD50108771 n/a 2000 n/a n/a n/a BindingDB BindingDB
84 MAP2K1 CHEMBL214752 BD50194054 n/a 2007 n/a 150 n/a BindingDB BindingDB
85 MAP2K1 CHEMBL201186 BD50176560 n/a 203 n/a n/a n/a BindingDB BindingDB
86 MAP2K1 CHEMBL215011 BD50194032 n/a 207 n/a 128 n/a BindingDB BindingDB
87 MAP2K1 CHEMBL282361 BD50099985 n/a 21 n/a n/a n/a BindingDB BindingDB
88 MAP2K1 CHEMBL485574 BD50274332 n/a 21 n/a n/a n/a BindingDB BindingDB
89 MAP2K1 CHEMBL95728 BD50072152 n/a 2100 n/a n/a n/a BindingDB BindingDB
90 MAP2K1 CHEMBL95057 BD50072158 n/a 2100 n/a n/a n/a BindingDB BindingDB
91 MAP2K1 CHEMBL330195 BD50072160 n/a 2100 n/a n/a n/a BindingDB BindingDB
92 MAP2K1 CHEMBL320688 BD50132267 n/a 212 n/a n/a n/a BindingDB BindingDB
93 MAP2K1 CHEMBL213651 BD50187812 n/a 220 n/a n/a n/a BindingDB BindingDB
94 MAP2K1 CHEMBL1169746 BD50321559 n/a 220 n/a n/a n/a BindingDB BindingDB
95 MAP2K1 CHEMBL203257 BD50180557 n/a 2200 n/a n/a n/a BindingDB BindingDB
96 MAP2K1 CHEMBL201389 BD50176569 n/a 23 n/a n/a n/a BindingDB BindingDB
97 MAP2K1 CHEMBL377288 BD50176595 n/a 23 n/a n/a n/a BindingDB BindingDB
98 MAP2K1 CHEMBL201246 BD50176577 n/a 2320 n/a n/a n/a BindingDB BindingDB
99 MAP2K1 CHEMBL202356 BD50176559 n/a 24 n/a n/a n/a BindingDB BindingDB
100 MAP2K1 CHEMBL253116 BD50196392 n/a 240 n/a 45 n/a BindingDB BindingDB
101 MAP2K1 CHEMBL524274 BD50265350 n/a 2400 n/a n/a n/a BindingDB BindingDB
102 MAP2K1 CHEMBL201203 BD50176581 n/a 241 n/a n/a n/a BindingDB BindingDB
103 MAP2K1 CHEMBL1288582 BD50331277 n/a 2450 n/a n/a n/a BindingDB BindingDB
104 MAP2K1 CHEMBL95002 BD50095235 n/a 25 n/a n/a n/a BindingDB BindingDB
105 MAP2K1 CHEMBL483398 BD50274386 n/a 25 n/a n/a n/a BindingDB BindingDB
106 MAP2K1 CHEMBL385820 BD50187815 n/a 250 n/a n/a n/a BindingDB BindingDB
107 MAP2K1 Debromohymenialdisine (DBH) BD00016591 n/a 2500 n/a n/a n/a BindingDB BindingDB
108 MAP2K1 CHEMBL356164 BD50108773 n/a 2500 n/a n/a n/a BindingDB BindingDB
109 MAP2K1 CHEMBL440356 BD50108774 n/a 2500 n/a n/a n/a BindingDB BindingDB
110 MAP2K1 CHEMBL359106 BD50108776 n/a 2500 n/a n/a n/a BindingDB BindingDB
111 MAP2K1 CHEMBL357047 BD50108777 n/a 2500 n/a n/a n/a BindingDB BindingDB
112 MAP2K1 CHEMBL151430 BD50108778 n/a 2500 n/a n/a n/a BindingDB BindingDB
113 MAP2K1 CHEMBL361708 BD50108779 n/a 2500 n/a n/a n/a BindingDB BindingDB
114 MAP2K1 CHEMBL397591 BD50220547 n/a 2500 n/a n/a n/a BindingDB BindingDB
115 MAP2K1 CHEMBL31497 BD50099988 n/a 26 n/a n/a n/a BindingDB BindingDB
116 MAP2K1 CHEMBL437331 BD50194024 n/a 26 n/a 42 n/a BindingDB BindingDB
117 MAP2K1 CHEMBL385446 BD50194030 n/a 26 n/a 220 n/a BindingDB BindingDB
118 MAP2K1 CHEMBL484368 BD50274245 n/a 26 n/a n/a n/a BindingDB BindingDB
119 MAP2K1 CHEMBL1684060 BD50337935 n/a 26 n/a n/a n/a BindingDB BindingDB
120 MAP2K1 CHEMBL95758 BD50072153 n/a 2600 n/a n/a n/a BindingDB BindingDB
121 MAP2K1 CHEMBL383098 BD50176579 n/a 2650 n/a n/a n/a BindingDB BindingDB
122 MAP2K1 CHEMBL387184 BD50194039 n/a 27 n/a 332 n/a BindingDB BindingDB
123 MAP2K1 CHEMBL214614 BD50194056 n/a 27 n/a >10 n/a BindingDB BindingDB
124 MAP2K1 CHEMBL321078 BD50132259 n/a 28 n/a n/a n/a BindingDB BindingDB
125 MAP2K1 CHEMBL385905 BD50194041 n/a 28 n/a 75 n/a BindingDB BindingDB
126 MAP2K1 CHEMBL30597 BD50099980 n/a 280 n/a n/a n/a BindingDB BindingDB
127 MAP2K1 CHEMBL217416 BD50194035 n/a 280 n/a 350 n/a BindingDB BindingDB
128 MAP2K1 CHEMBL97067 BD50072159 n/a 2800 n/a n/a n/a BindingDB BindingDB
129 MAP2K1 CHEMBL287852 BD50099976 n/a 29 n/a n/a n/a BindingDB BindingDB
130 MAP2K1 CHEMBL414856 BD50176593 n/a 29 n/a n/a n/a BindingDB BindingDB
131 MAP2K1 CHEMBL1171014 BD50321573 n/a 29 n/a n/a n/a BindingDB BindingDB
132 MAP2K1 CHEMBL386457 BD50194066 n/a 298 n/a 605 n/a BindingDB BindingDB
133 MAP2K1 3-cyanoquinoline, 3 BD00028118 n/a 3 n/a n/a n/a BindingDB BindingDB
134 MAP2K1 CHEMBL485615 BD50274438 n/a 3 n/a n/a n/a BindingDB BindingDB
135 MAP2K1 CHEMBL1684075 BD50337934 n/a 3.1 n/a n/a n/a BindingDB BindingDB
136 MAP2K1 CHEMBL1615025 BD50337926 n/a 3.2 n/a n/a n/a BindingDB BindingDB
137 MAP2K1 CHEMBL1684070 BD50337929 n/a 3.2 n/a n/a n/a BindingDB BindingDB
138 MAP2K1 CHEMBL1684074 BD50337933 n/a 3.3 n/a n/a n/a BindingDB BindingDB
139 MAP2K1 CHEMBL31806 BD50099990 n/a 3.6 n/a n/a n/a BindingDB BindingDB
140 MAP2K1 CHEMBL1684067 BD50337925 n/a 3.8 n/a n/a n/a BindingDB BindingDB
141 MAP2K1 CHEMBL199749 BD50180556 n/a 30 n/a n/a n/a BindingDB BindingDB
142 MAP2K1 CHEMBL203417 BD50180563 n/a 30 n/a n/a n/a BindingDB BindingDB
143 MAP2K1 CHEMBL269696 BD50194036 n/a 30 n/a >10 n/a BindingDB BindingDB
144 MAP2K1 CHEMBL215193 BD50194061 n/a 30 n/a 130 n/a BindingDB BindingDB
145 MAP2K1 CHEMBL485286 BD50264756 n/a 30 n/a n/a n/a BindingDB BindingDB
146 MAP2K1 CHEMBL1170191 BD50321575 n/a 30 n/a n/a n/a BindingDB BindingDB
147 MAP2K1 CHEMBL95069 BD50072154 n/a 300 n/a n/a n/a BindingDB BindingDB
148 MAP2K1 CHEMBL329492 BD50072163 n/a 300 n/a n/a n/a BindingDB BindingDB
149 MAP2K1 CHEMBL214901 BD50194051 n/a 32 n/a 47 n/a BindingDB BindingDB
150 MAP2K1 CHEMBL1171682 BD50321571 n/a 32 n/a n/a n/a BindingDB BindingDB
151 MAP2K1 CHEMBL95905 BD50072165 n/a 3200 n/a n/a n/a BindingDB BindingDB
152 MAP2K1 CHEMBL30551 BD50099991 n/a 33 n/a n/a n/a BindingDB BindingDB
153 MAP2K1 CHEMBL369992 BD50176592 n/a 33 n/a n/a n/a BindingDB BindingDB
154 MAP2K1 CHEMBL201426 BD50180573 n/a 33 n/a n/a n/a BindingDB BindingDB
155 MAP2K1 CHEMBL489661 BD50274437 n/a 33 n/a n/a n/a BindingDB BindingDB
156 MAP2K1 CHEMBL371969 BD50176602 n/a 331 n/a n/a n/a BindingDB BindingDB
157 MAP2K1 CHEMBL216449 BD50194023 n/a 34 n/a 65 n/a BindingDB BindingDB
158 MAP2K1 CHEMBL263039 BD50194026 n/a 34 n/a 22 n/a BindingDB BindingDB
159 MAP2K1 CHEMBL383858 BD50194031 n/a 34 n/a 113 n/a BindingDB BindingDB
160 MAP2K1 CHEMBL202128 BD50176587 n/a 3470 n/a n/a n/a BindingDB BindingDB
161 MAP2K1 CHEMBL97714 BD50095236 n/a 35 n/a n/a n/a BindingDB BindingDB
162 MAP2K1 CHEMBL216325 BD50194045 n/a 35 n/a 120 n/a BindingDB BindingDB
163 MAP2K1 CHEMBL519206 BD50274202 n/a 35 n/a n/a n/a BindingDB BindingDB
164 MAP2K1 CHEMBL377592 BD50187857 n/a 350 n/a n/a n/a BindingDB BindingDB
165 MAP2K1 CHEMBL378385 BD50176572 n/a 36 n/a n/a n/a BindingDB BindingDB
166 MAP2K1 CHEMBL485377 BD50274203 n/a 36 n/a n/a n/a BindingDB BindingDB
167 MAP2K1 CHEMBL201384 BD50176570 n/a 361 n/a n/a n/a BindingDB BindingDB
168 MAP2K1 CHEMBL215038 BD50194065 n/a 37 n/a 78 n/a BindingDB BindingDB
169 MAP2K1 CHEMBL375609 BD50187848 n/a 38 n/a 375 n/a BindingDB BindingDB
170 MAP2K1 CHEMBL201833 BD50176573 n/a 386 n/a n/a n/a BindingDB BindingDB
171 MAP2K1 CHEMBL201417 BD50180566 n/a 39 n/a n/a n/a BindingDB BindingDB
172 MAP2K1 CHEMBL202355 BD50176562 n/a 397 n/a n/a n/a BindingDB BindingDB
173 MAP2K1 3-cyanoquinoline, 4 BD00028119 n/a 4 n/a n/a n/a BindingDB BindingDB
174 MAP2K1 CHEMBL524111 BD50274439 n/a 4 n/a n/a n/a BindingDB BindingDB
175 MAP2K1 CHEMBL1684073 BD50337932 n/a 4 n/a n/a n/a BindingDB BindingDB
176 MAP2K1 CHEMBL30359 BD50099983 n/a 4.2 n/a n/a n/a BindingDB BindingDB
177 MAP2K1 CHEMBL288081 BD50099981 n/a 4.4 n/a n/a n/a BindingDB BindingDB
178 MAP2K1 CHEMBL1684063 BD50337920 n/a 4.6 n/a n/a n/a BindingDB BindingDB
179 MAP2K1 CHEMBL1684069 BD50337928 n/a 4.8 n/a n/a n/a BindingDB BindingDB
180 MAP2K1 CHEMBL1684062 BD50337937 n/a 4.9 n/a n/a n/a BindingDB BindingDB
181 MAP2K1 CHEMBL201630 BD50180571 n/a 40 n/a n/a n/a BindingDB BindingDB
182 MAP2K1 CHEMBL214587 BD50194034 n/a 40 n/a 35 n/a BindingDB BindingDB
183 MAP2K1 CHEMBL385059 BD50194046 n/a 40 n/a 694 n/a BindingDB BindingDB
184 MAP2K1 CHEMBL485285 BD50264755 n/a 40 n/a n/a n/a BindingDB BindingDB
185 MAP2K1 CHEMBL94971 BD50072166 n/a 400 n/a n/a n/a BindingDB BindingDB
186 MAP2K1 CHEMBL523559 BD50265034 n/a 400 n/a n/a n/a BindingDB BindingDB
187 MAP2K1 CHEMBL425065 BD50187829 n/a 410 n/a n/a n/a BindingDB BindingDB
188 MAP2K1 CHEMBL380328 BD50187852 n/a 410 n/a n/a n/a BindingDB BindingDB
189 MAP2K1 CHEMBL202063 BD50176586 n/a 42 n/a n/a n/a BindingDB BindingDB
190 MAP2K1 CHEMBL213992 BD50187817 n/a 42 n/a >10000 n/a BindingDB BindingDB
191 MAP2K1 CHEMBL1171312 BD50321563 n/a 42 n/a n/a n/a BindingDB BindingDB
192 MAP2K1 CHEMBL213563 BD50187830 n/a 420 n/a n/a n/a BindingDB BindingDB
193 MAP2K1 CHEMBL31384 BD50099982 n/a 43 n/a n/a n/a BindingDB BindingDB
194 MAP2K1 CHEMBL201156 BD50180570 n/a 43 n/a n/a n/a BindingDB BindingDB
195 MAP2K1 CHEMBL212110 BD50187850 n/a 430 n/a n/a n/a BindingDB BindingDB
196 MAP2K1 CHEMBL213167 BD50187818 n/a 44 n/a n/a n/a BindingDB BindingDB
197 MAP2K1 CHEMBL265478 BD50194016 n/a 44 n/a 140 n/a BindingDB BindingDB
198 MAP2K1 CHEMBL216832 BD50194063 n/a 44 n/a 49 n/a BindingDB BindingDB
199 MAP2K1 CHEMBL202771 BD50180565 n/a 4496 n/a n/a n/a BindingDB BindingDB
200 MAP2K1 CHEMBL199774 BD50180560 n/a 45 n/a n/a n/a BindingDB BindingDB
201 MAP2K1 CHEMBL386230 BD50194062 n/a 45 n/a 650 n/a BindingDB BindingDB
202 MAP2K1 CHEMBL330388 BD50095231 n/a 450 n/a n/a n/a BindingDB BindingDB
203 MAP2K1 CHEMBL97586 BD50072155 n/a 4500 n/a n/a n/a BindingDB BindingDB
204 MAP2K1 CHEMBL216833 BD50194028 n/a 46 n/a 47 n/a BindingDB BindingDB
205 MAP2K1 CHEMBL384012 BD50194055 n/a 46 n/a 54 n/a BindingDB BindingDB
206 MAP2K1 CHEMBL1169996 BD50321565 n/a 46 n/a n/a n/a BindingDB BindingDB
207 MAP2K1 CHEMBL265786 BD50176567 n/a 48 n/a n/a n/a BindingDB BindingDB
208 MAP2K1 CHEMBL97205 BD50072149 n/a 4800 n/a n/a n/a BindingDB BindingDB
209 MAP2K1 3-cyanoquinoline, 7 BD00028122 n/a 5 n/a n/a n/a BindingDB BindingDB
210 MAP2K1 CHEMBL520025 BD50274204 n/a 5 n/a n/a n/a BindingDB BindingDB
211 MAP2K1 CHEMBL1684071 BD50337930 n/a 5 n/a n/a n/a BindingDB BindingDB
212 MAP2K1 CHEMBL1681812 BD50337924 n/a 5.9 n/a n/a n/a BindingDB BindingDB
213 MAP2K1 CHEMBL317720 BD50072151 n/a 500 n/a n/a n/a BindingDB BindingDB
214 MAP2K1 CHEMBL378719 BD50187813 n/a 500 n/a n/a n/a BindingDB BindingDB
215 MAP2K1 CHEMBL212214 BD50187831 n/a 500 n/a n/a n/a BindingDB BindingDB
216 MAP2K1 CHEMBL378014 BD50187838 n/a 500 n/a n/a n/a BindingDB BindingDB
217 MAP2K1 CHEMBL209868 BD50187821 n/a 510 n/a 8321 n/a BindingDB BindingDB
218 MAP2K1 CHEMBL217414 BD50194059 n/a 52 n/a 88 n/a BindingDB BindingDB
219 MAP2K1 CHEMBL521320 BD50274244 n/a 52 n/a n/a n/a BindingDB BindingDB
220 MAP2K1 CHEMBL279758 BD50099972 n/a 520 n/a n/a n/a BindingDB BindingDB
221 MAP2K1 CHEMBL201716 BD50176566 n/a 521 n/a n/a n/a BindingDB BindingDB
222 MAP2K1 CHEMBL1684065 BD50337922 n/a 53 n/a n/a n/a BindingDB BindingDB
223 MAP2K1 CHEMBL217355 BD50194052 n/a 540 n/a 350 n/a BindingDB BindingDB
224 MAP2K1 CHEMBL201780 BD50176590 n/a 5420 n/a n/a n/a BindingDB BindingDB
225 MAP2K1 CHEMBL485211 BD50274243 n/a 55 n/a n/a n/a BindingDB BindingDB
226 MAP2K1 CHEMBL30268 BD50099973 n/a 550 n/a n/a n/a BindingDB BindingDB
227 MAP2K1 CHEMBL386469 BD50194019 n/a 56 n/a 444 n/a BindingDB BindingDB
228 MAP2K1 CHEMBL201302 BD50176599 n/a 566 n/a n/a n/a BindingDB BindingDB
229 MAP2K1 CHEMBL424897 BD50194033 n/a 57 n/a 250 n/a BindingDB BindingDB
230 MAP2K1 CHEMBL204535 BD50176564 n/a 58 n/a n/a n/a BindingDB BindingDB
231 MAP2K1 CHEMBL214683 BD50194025 n/a 58 n/a 43 n/a BindingDB BindingDB
232 MAP2K1 CHEMBL217310 BD50194050 n/a 58 n/a 130 n/a BindingDB BindingDB
233 MAP2K1 CHEMBL217832 BD50194058 n/a 58 n/a 123 n/a BindingDB BindingDB
234 MAP2K1 CHEMBL521013 BD50274242 n/a 59 n/a n/a n/a BindingDB BindingDB
235 MAP2K1 CHEMBL450271 BD50274440 n/a 6 n/a n/a n/a BindingDB BindingDB
236 MAP2K1 CHEMBL31733 BD50095226 n/a 6.2 n/a n/a n/a BindingDB BindingDB
237 MAP2K1 CHEMBL201629 BD50180564 n/a 6.8 n/a n/a n/a BindingDB BindingDB
238 MAP2K1 CHEMBL30763 BD50095239 n/a 60 n/a n/a n/a BindingDB BindingDB
239 MAP2K1 CHEMBL217415 BD50194022 n/a 60 n/a 330 n/a BindingDB BindingDB
240 MAP2K1 CHEMBL201200 BD50176594 n/a 6130 n/a n/a n/a BindingDB BindingDB
241 MAP2K1 CHEMBL211359 BD50187841 n/a 62 n/a 1480 n/a BindingDB BindingDB
242 MAP2K1 CHEMBL209845 BD50187827 n/a 620 n/a n/a n/a BindingDB BindingDB
243 MAP2K1 CHEMBL371658 BD50173838 n/a 630 n/a n/a n/a BindingDB BindingDB
244 MAP2K1 CHEMBL214816 BD50194057 n/a 64 n/a 140 n/a BindingDB BindingDB
245 MAP2K1 CHEMBL203414 BD50176578 n/a 642 n/a n/a n/a BindingDB BindingDB
246 MAP2K1 CHEMBL212305 BD50187835 n/a 650 n/a n/a n/a BindingDB BindingDB
247 MAP2K1 CHEMBL217126 BD50194064 n/a 67 n/a 70 n/a BindingDB BindingDB
248 MAP2K1 CHEMBL378688 BD50187856 n/a 670 n/a n/a n/a BindingDB BindingDB
249 MAP2K1 CHEMBL201136 BD50180559 n/a 6786 n/a n/a n/a BindingDB BindingDB
250 MAP2K1 CHEMBL94965 BD50095229 n/a 68 n/a n/a n/a BindingDB BindingDB
251 MAP2K1 CHEMBL202385 BD50176565 n/a 68 n/a n/a n/a BindingDB BindingDB
252 MAP2K1 CHEMBL377783 BD50187801 n/a 68 n/a n/a n/a BindingDB BindingDB
253 MAP2K1 CHEMBL98130 BD50095233 n/a 680 n/a n/a n/a BindingDB BindingDB
254 MAP2K1 CHEMBL209502 BD50187832 n/a 690 n/a n/a n/a BindingDB BindingDB
255 MAP2K1 CHEMBL1172521 BD50321576 n/a 7 n/a n/a n/a BindingDB BindingDB
256 MAP2K1 CHEMBL100473 BD50072147 n/a 70 n/a n/a n/a BindingDB BindingDB
257 MAP2K1 CHEMBL316510 BD50072148 n/a 700 n/a n/a n/a BindingDB BindingDB
258 MAP2K1 CHEMBL209793 BD50187849 n/a 7000 n/a n/a n/a BindingDB BindingDB
259 MAP2K1 CHEMBL1170596 BD50321560 n/a 72 n/a n/a n/a BindingDB BindingDB
260 MAP2K1 CHEMBL211201 BD50187855 n/a 73 n/a n/a n/a BindingDB BindingDB
261 MAP2K1 CHEMBL212480 BD50187822 n/a 740 n/a n/a n/a BindingDB BindingDB
262 MAP2K1 CHEMBL1684066 BD50337923 n/a 740 n/a n/a n/a BindingDB BindingDB
263 MAP2K1 CHEMBL216201 BD50194017 n/a 744 n/a 564 n/a BindingDB BindingDB
264 MAP2K1 CHEMBL214032 BD50194040 n/a 75 n/a 100 n/a BindingDB BindingDB
265 MAP2K1 CHEMBL202177 BD50176576 n/a 76 n/a n/a n/a BindingDB BindingDB
266 MAP2K1 CHEMBL491435 BD50264740 n/a 7600 n/a n/a n/a BindingDB BindingDB
267 MAP2K1 CHEMBL378833 BD50187858 n/a 790 n/a n/a n/a BindingDB BindingDB
268 MAP2K1 CHEMBL385703 BD50194018 n/a 7900 n/a 1500 n/a BindingDB BindingDB
269 MAP2K1 3-cyanoquinoline, 10 BD00028125 n/a 8 n/a n/a n/a BindingDB BindingDB
270 MAP2K1 CHEMBL1684064 BD50337921 n/a 8.3 n/a n/a n/a BindingDB BindingDB
271 MAP2K1 CHEMBL1684072 BD50337931 n/a 8.6 n/a n/a n/a BindingDB BindingDB
272 MAP2K1 CHEMBL214425 BD50194021 n/a 80 n/a 260 n/a BindingDB BindingDB
273 MAP2K1 CHEMBL371095 BD50173837 n/a 800 n/a n/a n/a BindingDB BindingDB
274 MAP2K1 CHEMBL212474 BD50187807 n/a 800 n/a n/a n/a BindingDB BindingDB
275 MAP2K1 CHEMBL204094 BD50176563 n/a 805 n/a n/a n/a BindingDB BindingDB
276 MAP2K1 CHEMBL203138 BD50180569 n/a 82 n/a n/a n/a BindingDB BindingDB
277 MAP2K1 CHEMBL215012 BD50194037 n/a 85 n/a 250 n/a BindingDB BindingDB
278 MAP2K1 CHEMBL213168 BD50187845 n/a 86 n/a n/a n/a BindingDB BindingDB
279 MAP2K1 CHEMBL201819 BD50176571 n/a 87 n/a n/a n/a BindingDB BindingDB
280 MAP2K1 CHEMBL102786 BD50132263 n/a 9 n/a n/a n/a BindingDB BindingDB
281 MAP2K1 CHEMBL372600 BD50180558 n/a 9.3 n/a n/a n/a BindingDB BindingDB
282 MAP2K1 CHEMBL1684061 BD50337936 n/a 9.8 n/a n/a n/a BindingDB BindingDB
283 MAP2K1 CHEMBL1169998 BD50321569 n/a 90 n/a n/a n/a BindingDB BindingDB
284 MAP2K1 CHEMBL330393 BD50072156 n/a 900 n/a n/a n/a BindingDB BindingDB
285 MAP2K1 CHEMBL97406 BD50072162 n/a 900 n/a n/a n/a BindingDB BindingDB
286 MAP2K1 CHEMBL329698 BD50072164 n/a 900 n/a n/a n/a BindingDB BindingDB
287 MAP2K1 CHEMBL380765 BD50176603 n/a 94 n/a n/a n/a BindingDB BindingDB
288 MAP2K1 CHEMBL199210 BD50173833 n/a 960 n/a n/a n/a BindingDB BindingDB
289 MAP2K1 CHEMBL1762110 BD50340954 n/a 960 n/a n/a n/a BindingDB BindingDB
290 MAP2K1 CHEMBL496536 BD50265308 n/a 9700 n/a n/a n/a BindingDB BindingDB
291 MAP2K1 CHEMBL30516 BD50099989 n/a 99 n/a n/a n/a BindingDB BindingDB
292 MAP2K1 CHEBI:305251 BD50117315 n/a <1 n/a n/a n/a BindingDB BindingDB
293 MAP2K1 CHEMBL1614766 BD50338038 n/a n/a 0.24 n/a n/a BindingDB BindingDB
294 MAP2K1 CHEMBL507361 BD50338039 n/a n/a 0.4 n/a n/a BindingDB BindingDB
295 MAP2K1 BIBF_1120der BIBF_1120der n/a n/a 10 n/a n/a NB2011DRx NB2011DRx
296 MAP2K1 BMS-354825 BD00013216 n/a n/a 1000 n/a n/a BindingDB BindingDB
297 MAP2K1 Dasatinib Dasatinib n/a n/a 1000 n/a n/a NB2008 NB2008
298 MAP2K1 Dasatinib Dasatinib n/a n/a 1000 n/a n/a NB2011DRx NB2011DRx
299 MAP2K1 PHA_665752 PHA_665752 n/a n/a 1100 n/a n/a NB2011DRx NB2011DRx
300 MAP2K1 EXEL_2880 EXEL_2880 n/a n/a 12 n/a n/a NB2011DRx NB2011DRx
301 MAP2K1 CI_1040 CI_1040 n/a n/a 120 n/a n/a NB2011DRx NB2011DRx
302 MAP2K1 SU11248 BD00004814 n/a n/a 130 n/a n/a BindingDB BindingDB
303 MAP2K1 Sunitinib Sunitinib n/a n/a 130 n/a n/a NB2008 NB2008
304 MAP2K1 Sunitinib Sunitinib n/a n/a 130 n/a n/a NB2011DRx NB2011DRx
305 MAP2K1 HKI_272 HKI_272 n/a n/a 14 n/a n/a NB2011DRx NB2011DRx
306 MAP2K1 Ki_20227 Ki_20227 n/a n/a 1700 n/a n/a NB2011DRx NB2011DRx
307 MAP2K1 VX-680 BD00013534 n/a n/a 1800 n/a n/a BindingDB BindingDB
308 MAP2K1 ZD6474 BD00004655 n/a n/a 1800 n/a n/a BindingDB BindingDB
309 MAP2K1 CI-1033 BD00004779 n/a n/a 1800 n/a n/a BindingDB BindingDB
310 MAP2K1 JNJ-7706621 BD00006866 n/a n/a 1800 n/a n/a BindingDB BindingDB
311 MAP2K1 CI_1033 CI_1033 n/a n/a 1800 n/a n/a NB2008 NB2008
312 MAP2K1 CI_1033 CI_1033 n/a n/a 1800 n/a n/a NB2011DRx NB2011DRx
313 MAP2K1 JNJ_7706621 JNJ_7706621 n/a n/a 1800 n/a n/a NB2008 NB2008
314 MAP2K1 Vandetanib Vandetanib n/a n/a 1800 n/a n/a NB2011DRx NB2011DRx
315 MAP2K1 VX_680 VX_680 n/a n/a 1800 n/a n/a NB2008 NB2008
316 MAP2K1 VX_680 VX_680 n/a n/a 1800 n/a n/a NB2011DRx NB2011DRx
317 MAP2K1 ZD_6474 ZD_6474 n/a n/a 1800 n/a n/a NB2008 NB2008
318 MAP2K1 SKI_606 SKI_606 n/a n/a 19 n/a n/a NB2011DRx NB2011DRx
319 MAP2K1 AZD_1152HQPA AZD_1152HQPA n/a n/a 1900 n/a n/a NB2011DRx NB2011DRx
320 MAP2K1 INCB18424 INCB18424 n/a n/a 1900 n/a n/a NB2011DRx NB2011DRx
321 MAP2K1 JNJ_28312141 JNJ_28312141 n/a n/a 200 n/a n/a NB2011DRx NB2011DRx
322 MAP2K1 Staurosporine Staurosporine n/a n/a 21 n/a n/a NB2008 NB2008
323 MAP2K1 Staurosporine Staurosporine n/a n/a 21 n/a n/a NB2011DRx NB2011DRx
324 MAP2K1 AG_013736 AG_013736 n/a n/a 2700 n/a n/a NB2011DRx NB2011DRx
325 MAP2K1 CHEMBL603469 BD50308060 n/a n/a 3.5 n/a n/a BindingDB BindingDB
326 MAP2K1 CEP_701 CEP_701 n/a n/a 3.5 n/a n/a NB2011DRx NB2011DRx
327 MAP2K1 R406 R406 n/a n/a 320 n/a n/a NB2011DRx NB2011DRx
328 MAP2K1 CHEBI:259924 BD50119072 n/a n/a 360 n/a n/a BindingDB BindingDB
329 MAP2K1 EKB_569 EKB_569 n/a n/a 360 n/a n/a NB2008 NB2008
330 MAP2K1 PP_242 PP_242 n/a n/a 51 n/a n/a NB2011DRx NB2011DRx
331 MAP2K1 TG_101348 TG_101348 n/a n/a 5100 n/a n/a NB2011DRx NB2011DRx
332 MAP2K1 CHEMBL522892 BD50265677 n/a n/a 520 n/a n/a BindingDB BindingDB
333 MAP2K1 CHIR_258 CHIR_258 n/a n/a 520 n/a n/a NB2008 NB2008
334 MAP2K1 CHIR_258 CHIR_258 n/a n/a 520 n/a n/a NB2011DRx NB2011DRx
335 MAP2K1 KW_2449 KW_2449 n/a n/a 530 n/a n/a NB2011DRx NB2011DRx
336 MAP2K1 PLX_4720 PLX_4720 n/a n/a 550 n/a n/a NB2011DRx NB2011DRx
337 MAP2K1 TAE_684 TAE_684 n/a n/a 550 n/a n/a NB2011DRx NB2011DRx
338 MAP2K1 cid_10138259 BD00031095 n/a n/a 77 n/a n/a BindingDB BindingDB
339 MAP2K1 SU_14813 SU_14813 n/a n/a 77 n/a n/a NB2008 NB2008
340 MAP2K1 SU_14813 SU_14813 n/a n/a 77 n/a n/a NB2011DRx NB2011DRx
341 MAP2K1 PD_173955 PD_173955 n/a n/a 830 n/a n/a NB2011DRx NB2011DRx
342 MAP2K1 AZD_6244 AZD_6244 n/a n/a 99 n/a n/a NB2011DRx NB2011DRx
343 MAP2K1 3BM 3BM n/a n/a n/a n/a n/a PDB PDB
344 MAP2K1 ADP ADP n/a n/a n/a n/a n/a PDB PDB
345 MAP2K1 AGS AGS n/a n/a n/a n/a n/a PDB PDB
346 MAP2K1 ANP ANP n/a n/a n/a n/a n/a PDB PDB
347 MAP2K1 ATP ATP n/a n/a n/a n/a n/a PDB PDB
348 MAP2K1 CAS135897_06_2 CAS135897_06_2 n/a n/a n/a n/a 29.48 NB2011RBC NB2011RBC
349 MAP2K1 CAS326914_10_7 CAS326914_10_7 n/a n/a n/a n/a 33.08 NB2011RBC NB2011RBC
350 MAP2K1 CAS62996_74_1 CAS62996_74_1 n/a n/a n/a n/a 3.83 NB2011RBC NB2011RBC
351 MAP2K1 CAS97161_97_2 CAS97161_97_2 n/a n/a n/a n/a 23.65 NB2011RBC NB2011RBC
352 MAP2K1 KSA KSA n/a n/a n/a n/a n/a PDB PDB