Query kinase |
SRPK2 (P78362)
|
Kinase group |
CMGC |
Number of inhibitors |
33 |
Index |
Target |
Inhibitor |
Inhibitor 2D |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
POC |
Source |
Link |
0 |
SRPK2 |
TG_101348 |
TG_101348 |
n/a |
n/a |
100 |
n/a |
n/a |
NB2011DRx |
NB2011DRx |
1 |
SRPK2 |
A_674563 |
A_674563 |
n/a |
n/a |
1100 |
n/a |
n/a |
NB2011DRx |
NB2011DRx |
2 |
SRPK2 |
LY_333531 |
LY_333531 |
n/a |
n/a |
1100 |
n/a |
n/a |
NB2011DRx |
NB2011DRx |
3 |
SRPK2 |
KW_2449 |
KW_2449 |
n/a |
n/a |
15 |
n/a |
n/a |
NB2011DRx |
NB2011DRx |
4 |
SRPK2 |
SU11248 |
BD00004814 |
n/a |
n/a |
190 |
n/a |
n/a |
BindingDB |
BindingDB |
5 |
SRPK2 |
Sunitinib |
Sunitinib |
n/a |
n/a |
190 |
n/a |
n/a |
NB2008 |
NB2008 |
6 |
SRPK2 |
Sunitinib |
Sunitinib |
n/a |
n/a |
190 |
n/a |
n/a |
NB2011DRx |
NB2011DRx |
7 |
SRPK2 |
cid_10138259 |
BD00031095 |
n/a |
n/a |
200 |
n/a |
n/a |
BindingDB |
BindingDB |
8 |
SRPK2 |
SU_14813 |
SU_14813 |
n/a |
n/a |
200 |
n/a |
n/a |
NB2008 |
NB2008 |
9 |
SRPK2 |
SU_14813 |
SU_14813 |
n/a |
n/a |
200 |
n/a |
n/a |
NB2011DRx |
NB2011DRx |
10 |
SRPK2 |
JNJ_28312141 |
JNJ_28312141 |
n/a |
n/a |
2200 |
n/a |
n/a |
NB2011DRx |
NB2011DRx |
11 |
SRPK2 |
CHEMBL522892 |
BD50265677 |
n/a |
n/a |
290 |
n/a |
n/a |
BindingDB |
BindingDB |
12 |
SRPK2 |
CHIR_258 |
CHIR_258 |
n/a |
n/a |
290 |
n/a |
n/a |
NB2008 |
NB2008 |
13 |
SRPK2 |
CHIR_258 |
CHIR_258 |
n/a |
n/a |
290 |
n/a |
n/a |
NB2011DRx |
NB2011DRx |
14 |
SRPK2 |
CHEBI:668343 |
BD50298227 |
n/a |
n/a |
330 |
n/a |
n/a |
BindingDB |
BindingDB |
15 |
SRPK2 |
CHEMBL608533 |
BD50326053 |
n/a |
n/a |
330 |
n/a |
n/a |
BindingDB |
BindingDB |
16 |
SRPK2 |
PKC_412 |
PKC_412 |
n/a |
n/a |
330 |
n/a |
n/a |
NB2008 |
NB2008 |
17 |
SRPK2 |
PKC_412 |
PKC_412 |
n/a |
n/a |
330 |
n/a |
n/a |
NB2011DRx |
NB2011DRx |
18 |
SRPK2 |
BIBF_1120der |
BIBF_1120der |
n/a |
n/a |
36 |
n/a |
n/a |
NB2011DRx |
NB2011DRx |
19 |
SRPK2 |
PHA_665752 |
PHA_665752 |
n/a |
n/a |
500 |
n/a |
n/a |
NB2011DRx |
NB2011DRx |
20 |
SRPK2 |
CHEMBL603469 |
BD50308060 |
n/a |
n/a |
51 |
n/a |
n/a |
BindingDB |
BindingDB |
21 |
SRPK2 |
CEP_701 |
CEP_701 |
n/a |
n/a |
51 |
n/a |
n/a |
NB2011DRx |
NB2011DRx |
22 |
SRPK2 |
CHEMBL162 |
BD50059889 |
n/a |
n/a |
67 |
n/a |
n/a |
BindingDB |
BindingDB |
23 |
SRPK2 |
Staurosporine |
Staurosporine |
n/a |
n/a |
67 |
n/a |
n/a |
NB2008 |
NB2008 |
24 |
SRPK2 |
Staurosporine |
Staurosporine |
n/a |
n/a |
67 |
n/a |
n/a |
NB2011DRx |
NB2011DRx |
25 |
SRPK2 |
VX-680 |
BD00013534 |
n/a |
n/a |
680 |
n/a |
n/a |
BindingDB |
BindingDB |
26 |
SRPK2 |
VX_680 |
VX_680 |
n/a |
n/a |
680 |
n/a |
n/a |
NB2008 |
NB2008 |
27 |
SRPK2 |
VX_680 |
VX_680 |
n/a |
n/a |
680 |
n/a |
n/a |
NB2011DRx |
NB2011DRx |
28 |
SRPK2 |
CAS212779_48_1 |
CAS212779_48_1 |
n/a |
n/a |
n/a |
n/a |
37.05 |
NB2011RBC |
NB2011RBC |
29 |
SRPK2 |
CAS220792_57_4 |
CAS220792_57_4 |
n/a |
n/a |
n/a |
n/a |
30.98 |
NB2011RBC |
NB2011RBC |
30 |
SRPK2 |
CAS443798_55_8 |
CAS443798_55_8 |
n/a |
n/a |
n/a |
n/a |
17.1 |
NB2011RBC |
NB2011RBC |
31 |
SRPK2 |
CAS62996_74_1 |
CAS62996_74_1 |
n/a |
n/a |
n/a |
n/a |
40.95 |
NB2011RBC |
NB2011RBC |
32 |
SRPK2 |
PVB |
PVB |
n/a |
n/a |
n/a |
n/a |
n/a |
PDB |
PDB |
|
|