Kinase profiling results of kinases in KIF 1H07A_MFP (CDK2, PDB code: 1H07, chain A)
Template Kinase: CDK2
Template inhibitor: AC1NAKJQ

90 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C C C C C C
ROCK1AGC      
ROCK2AGC      
GRK4AGC      
GRK7AGC      
MAST1AGC      
PRKCDAGC      
PRKCQAGC      
PRKCEAGC      
PKN1AGC      
PKN2AGC      
CAMK2ACAMK      
CHEK1CAMK      
CASKCAMK      
DCLK3CAMK      
PHKG1CAMK      
PHKG2CAMK      
PRKD1CAMK      
PRKD2CAMK      
PRKD3CAMK      
CHEK2CAMK      
CDK2CMGC      
CDK4CMGC      
CDK7CMGC      
PCTK1CMGC      
CDK15CMGC      
PFTK1CMGC      
CLK1CMGC      
CLK2CMGC      
CLK3CMGC      
CLK4CMGC      
HIPK1CMGC      
HIPK2CMGC      
HIPK3CMGC      
HIPK4CMGC      
MAPK7CMGC      
NLKCMGC      
MAPK14CMGC      
CAMKK2Other      
GAKOther      
NEK1Other      
NEK11Other      
NEK2Other      
NEK4Other      
STK35Other      
PLK1Other      
PLK2Other      
TLK2Other      
STK36Other      
STK39STE      
PAK1STE      
PAK2STE      
PAK3STE      
SLKSTE      
STK24STE      
MAP2K1STE      
MAP2K4STE      
MAP2K5STE      
ABL1TK      
TNK2TK      
AXLTK      
DDR1TK      
DDR2TK      
EPHA1TK      
EPHB1TK      
EPHB3TK      
PTK2TK      
FERTK      
FESTK      
FGFR2TK      
JAK2TK      
JAK3TK      
METTK      
MST1RTK      
FGRTK      
FYNTK      
SRCTK      
YES1TK      
BLKTK      
HCKTK      
LCKTK      
SRMSTK      
ZAP70TK      
BMXTK      
ITKTK      
NTRK2TK      
NTRK3TK      
IRAK4TKL      
TNNI3KTKL      
MAP3K7TKL      

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C
GRK4AGC   
GRK7AGC   
PKN1AGC   
PKN2AGC   
PRKCAAGC   
PRKCDAGC   
PRKCEAGC   
PRKCQAGC   
ROCK1AGC   
ROCK2AGC   
CAMK2ACAMK   
CHEK1CAMK   
CHEK2CAMK   
PHKG1CAMK   
PHKG2CAMK   
PRKD1CAMK   
PRKD2CAMK   
PRKD3CAMK   
CDK2CMGC   
CDK4CMGC   
CDK7CMGC   
CLK1CMGC   
CLK2CMGC   
CLK3CMGC   
CLK4CMGC   
HIPK1CMGC   
HIPK2CMGC   
HIPK3CMGC   
HIPK4CMGC   
MAPK14CMGC   
NLKCMGC   
CAMKK2Other   
NEK1Other   
NEK11Other   
NEK2Other   
NEK4Other   
PLK1Other   
PLK2Other   
TLK2Other   
MAP2K1STE   
PAK1STE   
PAK2STE   
PAK3STE   
SLKSTE   
STK24STE   
STK39STE   
ABL1TK   
AXLTK   
BLKTK   
BMXTK   
DDR2TK   
EPHA1TK   
EPHB1TK   
EPHB3TK   
FERTK   
FESTK   
FGFR2TK   
FGRTK   
FYNTK   
HCKTK   
ITKTK   
JAK2TK   
JAK3TK   
LCKTK   
METTK   
MST1RTK   
NTRK2TK   
NTRK3TK   
PTK2TK   
SRCTK   
SRMSTK   
TNK2TK   
YES1TK   
ZAP70TK   
IRAK4TKL   
MAP3K7TKL