Kinase profiling results of kinases in KIF 2WIHA_P48 (CDK2, PDB code: 2WIH, chain A)
Template Kinase: CDK2
Template inhibitor: VX_680

111 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C C C C C C C C
AKT1AGC        
AKT2AGC        
ROCK1AGC        
GRK4AGC        
PDPK1AGC        
PRKCDAGC        
PRKCQAGC        
PKN1AGC        
PKN2AGC        
RPS6KA1AGC        
RPS6KA1CAMK        
RPS6KA2AGC        
RPS6KA2CAMK        
RPS6KA3AGC        
CAMK1GCAMK        
BRSK1CAMK        
CHEK1CAMK        
HUNKCAMK        
MARK1CAMK        
MARK2CAMK        
MARK3CAMK        
MARK4CAMK        
NUAK1CAMK        
NUAK2CAMK        
SIK1CAMK        
SIK2CAMK        
STK33CAMK        
DAPK3CAMK        
STK17ACAMK        
PHKG1CAMK        
PHKG2CAMK        
CDK2CMGC        
CDK4CMGC        
CDK5CMGC        
CDK9CMGC        
PCTK1CMGC        
PCTK2CMGC        
CDK11ACMGC        
CDK11ACMGC        
CDKL2CMGC        
CDKL3CMGC        
CDKL5CMGC        
CSNK2A1CMGC        
CSNK2A2CMGC        
PRPF4BCMGC        
GSK3ACMGC        
GSK3BCMGC        
MAPK10CMGC        
MAPK8CMGC        
MAPK14CMGC        
AURKAOther        
AURKBOther        
AURKCOther        
CAMKK1Other        
CHUKOther        
NEK5Other        
PLK1Other        
PLK2Other        
PLK3Other        
TTKOther        
ULK3Other        
PAK1STE        
PAK2STE        
PAK3STE        
SLKSTE        
STK10STE        
STK24STE        
STK25STE        
MAP2K1STE        
MAP2K6STE        
MAP2K5STE        
ABL1TK        
ABL2TK        
TNK2TK        
AXLTK        
DDR1TK        
DDR2TK        
EPHB1TK        
FERTK        
FESTK        
FGFR1TK        
FGFR2TK        
FGFR3TK        
FGFR4TK        
JAK1TK        
JAK2TK        
JAK3TK        
METTK        
MUSKTK        
FRKTK        
FGRTK        
FYNTK        
SRCTK        
YES1TK        
BLKTK        
HCKTK        
LCKTK        
LYNTK        
PTK6TK        
BMXTK        
ITKTK        
NTRK2TK        
NTRK3TK        
IRAK4TKL        
TESK1TKL        
MAP3K12TKL        
MAP3K13TKL        
MAP3K10TKL        
MAP3K11TKL        
MAP3K9TKL        
MAP3K7TKL        
ZAKTKL        

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C C C C C C
AKT1AGC         
AKT2AGC         
GRK4AGC         
PDPK1AGC         
PKN1AGC         
PKN2AGC         
PRKCAAGC         
PRKCDAGC         
PRKCQAGC         
ROCK1AGC         
RPS6KA1AGC         
RPS6KA2AGC         
RPS6KA3AGC         
BRSK1CAMK         
CAMK1GCAMK         
CHEK1CAMK         
DAPK3CAMK         
MARK1CAMK         
MARK2CAMK         
MARK3CAMK         
MARK4CAMK         
NUAK1CAMK         
NUAK2CAMK         
PHKG1CAMK         
PHKG2CAMK         
SIK2CAMK         
STK17ACAMK         
STK33CAMK         
CDC2CMGC         
CDC2CMGC         
CDK2CMGC         
CDK4CMGC         
CDK5CMGC         
CDK9CMGC         
CSNK2A1CMGC         
CSNK2A2CMGC         
GSK3ACMGC         
GSK3BCMGC         
MAPK10CMGC         
MAPK14CMGC         
MAPK8CMGC         
AURKAOther         
AURKBOther         
AURKCOther         
CAMKK1Other         
CHUKOther         
PLK1Other         
PLK2Other         
PLK3Other         
TTKOther         
ULK3Other         
MAP2K1STE         
MAP2K6STE         
PAK1STE         
PAK2STE         
PAK3STE         
SLKSTE         
STK10STE         
STK24STE         
STK25STE         
ABL1TK         
ABL2TK         
AXLTK         
BLKTK         
BMXTK         
DDR2TK         
EPHB1TK         
FERTK         
FESTK         
FGFR1TK         
FGFR2TK         
FGFR3TK         
FGFR4TK         
FGRTK         
FRKTK         
FYNTK         
HCKTK         
ITKTK         
JAK1TK         
JAK2TK         
JAK3TK         
LCKTK         
LYNTK         
METTK         
MUSKTK         
NTRK2TK         
NTRK3TK         
PTK6TK         
SRCTK         
TNK2TK         
YES1TK         
IRAK4TKL         
MAP3K10TKL         
MAP3K11TKL         
MAP3K7TKL         
MAP3K9TKL         
ZAKTKL