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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
CDKL3 (
Q8IVW4
)
Kinase group
CMGC
Number of conformation types
0
Number of structural templates
28 (
Total 10 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
20
2HZ4A_4ST
(ABL1)
CMGC
staurosporine
I
159
103
156
A
2HZ4A_4ST
(ABL1)
CMGC
staurosporine
I
159
103
156
159
103
156
A
2F4JA_VX6
(ABL1)
CMGC
VX-680
I
110
109
134
110
109
134
A
3A4OX_STU
(LYN)
CMGC
staurosporine
I
73
70
88
73
70
88
A
2WIHA_P48
(CDK2)
CMGC
VX_680
I
111
425
105
111
425
105
A
2JDRA_L20
(AKT2)
CMGC
A-443654
I
44
255
61
44
255
61
A
1PKDA_UCN
(CDK2)
CMGC
UCN 02
I
195
67
118
195
67
118
A
2XYNA_VX6
(ABL2)
CMGC
VX-680
I
79
101
105
79
101
105
A
1AQ1A_STU
(CDK2)
CMGC
staurosporine
I
195
76
118
195
76
118
A
1Q3DA_STU
(GSK3B)
CMGC
staurosporine
I
115
71
61
115
71
61
A
3E5AA_VX6
(AURKA)
CMGC
VX-680
I
57
107
93
57
107
93
A
1BYGA_STU
(CSK)
CMGC
staurosporine
I
85
72
123
85
72
123
A
1XJDA_STU
(PRKCQ)
CMGC
staurosporine
I
121
101
106
121
101
106
A
1NVQA_UCN
(CHEK1)
CMGC
UCN 02
I
179
65
79
179
65
79
A
1YHSA_STU
(PIM1)
CMGC
staurosporine
I
78
64
50
78
64
50
A
3CKXA_STU
(STK24)
CMGC
staurosporine
I
176
104
141
176
104
141
A
1NVRA_STU
(CHEK1)
CMGC
staurosporine
I
179
71
79
179
71
79
A
1YVJA_4ST
(JAK3)
CMGC
staurosporine
I
96
90
126
96
90
126
A
1NXKA_STU
(MAPKAPK2)
CMGC
staurosporine
I
110
67
51
110
67
51
A
2HY81_1ST
(PAK1)
CMGC
UCN 02
I
58
20
75
58
20
75
A
3FMEA_STU
(MAP2K6)
CMGC
staurosporine
I
28
15
20
28
15
20
B
8
3NYNA_SGV
(GRK6)
CMGC
SMR000127424
I
54
7
47
B
3NYNA_SGV
(GRK6)
CMGC
SMR000127424
I
54
7
47
54
7
47
B
1OKYA_STU
(PDPK1)
CMGC
staurosporine
I
179
67
109
179
67
109
B
3EFWA_AK8
(AURKA)
CMGC
3efw
I
100
59
105
100
59
105
B
1OKZA_UCN
(PDPK1)
CMGC
UCN 02
I
179
60
109
179
60
109
B
3BKBA_STU
(FES)
CMGC
staurosporine
I
131
107
138
131
107
138
B
3CBLA_STU
(FES)
CMGC
staurosporine
I
131
107
138
131
107
138
B
3CD3A_STU
(FES)
CMGC
staurosporine
I
131
107
138
131
107
138
B
3D7TA_STU
(CSK)
CMGC
staurosporine
I
70
68
99
70
68
99