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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
MAP2K5 (
Q13163
)
Kinase group
STE
Number of conformation types
0
Number of structural templates
29 (
Total 43 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
27
2H8HA_H8H
(SRC)
STE
Saracatinib
I
91
255
126
A
2H8HA_H8H
(SRC)
STE
Saracatinib
I
91
255
126
91
255
126
A
3EQFA_KSA
(MAP2K1)
STE
k-252a
I
42
51
57
42
51
57
A
2OW3A_BIM
(GSK3B)
STE
LY_333531
I
62
139
51
62
139
51
A
1AQ1A_STU
(CDK2)
STE
staurosporine
I
195
76
118
195
76
118
A
3CKXA_STU
(STK24)
STE
staurosporine
I
176
104
141
176
104
141
A
2GQGA_1N1
(ABL1)
STE
Dasatinib
I
74
32
117
74
32
117
A
1OPLA_P16
(ABL1)
STE
PD166326
I
89
70
123
89
70
123
A
1NVQA_UCN
(CHEK1)
STE
UCN 02
I
179
65
79
179
65
79
A
2VTTA_LZD
(CDK2)
STE
pyrazole dia...
I
158
42
111
158
42
111
A
1M17A_AQ4
(EGFR)
STE
Erlotinib
I
43
166
82
43
166
82
A
2FO0A_P16
(ABL1)
STE
PD166326
I
89
70
123
89
70
123
A
1NVRA_STU
(CHEK1)
STE
staurosporine
I
179
71
79
179
71
79
A
1R78A_FMD
(CDK2)
STE
4-alkynyl ox...
I
127
24
97
127
24
97
A
1OI9A_N20
(CDK2)
STE
NU-6086
I
52
80
61
52
80
61
A
2G2HA_P16
(ABL1)
STE
PD166326
I
89
70
123
89
70
123
A
1PKDA_UCN
(CDK2)
STE
UCN 02
I
195
67
118
195
67
118
A
2F4JA_VX6
(ABL1)
STE
VX-680
I
110
109
134
110
109
134
A
2HZIA_JIN
(ABL1)
STE
PD180970
I
90
77
120
90
77
120
A
1Q3DA_STU
(GSK3B)
STE
staurosporine
I
115
71
61
115
71
61
A
2WIHA_P48
(CDK2)
STE
VX_680
I
111
425
105
111
425
105
A
3IKAA_0UN
(EGFR)
STE
2jkk
I
76
120
108
76
120
108
A
1SM2A_STU
(ITK)
STE
staurosporine
I
99
104
128
99
104
128
A
1XKKA_FMM
(EGFR)
STE
Lapatinib
I
9
79
31
9
79
31
A
1SNUA_STU
(ITK)
STE
staurosporine
I
99
104
128
99
104
128
A
3BBTB_FMM
(ERBB4)
STE
Lapatinib
I
9
79
31
9
79
31
A
2IW6A_QQ2
(CDK2)
STE
2iw6
I
112
209
86
112
209
86
A
2HZ4A_4ST
(ABL1)
STE
staurosporine
I
159
103
156
159
103
156
B
2
1H00A_FAP
(CDK2)
STE
AC1NAE4F
I
50
94
75
B
1H00A_FAP
(CDK2)
STE
AC1NAE4F
I
50
94
75
50
94
75
B
1H07A_MFP
(CDK2)
STE
AC1NAKJQ
I
90
241
80
90
241
80