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Example2
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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
1 PKN2 related diseases
hsa05132
Salmonella infection
Summary of query kinase
Query kinase
PKN2 (
Q16513
)
Kinase group
AGC
Number of conformation types
0
Number of structural templates
65 (
Total 57 inhibitors
)
Number of PKN2 related diseases
1 (
hsa05132
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
44
1PKDA_UCN
(CDK2)
AGC
UCN 02
I
195
67
118
A
1PKDA_UCN
(CDK2)
AGC
UCN 02
I
195
67
118
195
67
118
A
2DQ7X_STU
(FYN)
AGC
staurosporine
I
91
74
124
91
74
124
A
1AQ1A_STU
(CDK2)
AGC
staurosporine
I
195
76
118
195
76
118
A
1Q3DA_STU
(GSK3B)
AGC
staurosporine
I
115
71
61
115
71
61
A
2HW7A_STU
(MKNK2)
AGC
staurosporine
I
28
55
16
28
55
16
A
1BYGA_STU
(CSK)
AGC
staurosporine
I
85
72
123
85
72
123
A
1SM2A_STU
(ITK)
AGC
staurosporine
I
99
104
128
99
104
128
A
2HZ4A_4ST
(ABL1)
AGC
staurosporine
I
159
103
156
159
103
156
A
1NVQA_UCN
(CHEK1)
AGC
UCN 02
I
179
65
79
179
65
79
A
1SNUA_STU
(ITK)
AGC
staurosporine
I
99
104
128
99
104
128
A
1NVRA_STU
(CHEK1)
AGC
staurosporine
I
179
71
79
179
71
79
A
1U59A_STU
(ZAP70)
AGC
staurosporine
I
96
80
114
96
80
114
A
1NXKA_STU
(MAPKAPK2)
AGC
staurosporine
I
110
67
51
110
67
51
A
1XJDA_STU
(PRKCQ)
AGC
staurosporine
I
121
101
106
121
101
106
A
3CKXA_STU
(STK24)
AGC
staurosporine
I
176
104
141
176
104
141
A
1YVJA_4ST
(JAK3)
AGC
staurosporine
I
96
90
126
96
90
126
A
2XIKA_J60
(STK25)
AGC
SU11652
I
59
49
65
59
49
65
A
2VTTA_LZD
(CDK2)
AGC
pyrazole dia...
I
158
42
111
158
42
111
A
2J51A_DKI
(SLK)
AGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2I0EA_PDS
(PRKCB)
AGC
bisindolylma...
I
41
141
45
41
141
45
A
3M2WA_L8I
(MAPKAPK2)
AGC
Sunitinib
I
84
90
47
84
90
47
A
2JFLA_DKI
(SLK)
AGC
5-AMINO-3-{[...
I
90
11
103
90
11
103
A
2OW3A_BIM
(GSK3B)
AGC
LY_333531
I
62
139
51
62
139
51
A
2VD5A_BI8
(DMPK)
AGC
Ro 31-7549
I
19
49
12
19
49
12
A
3IW4A_LW4
(PRKCA)
AGC
Sotrastaurin
I
52
119
49
52
119
49
A
1R78A_FMD
(CDK2)
AGC
4-alkynyl ox...
I
127
24
97
127
24
97
A
2ETRA_Y27
(ROCK1)
AGC
y-27632
I
3
6
3
3
6
3
A
2CKEA_IQU
(DAPK2)
AGC
AEIQS
I
10
17
22
10
17
22
A
3E5AA_VX6
(AURKA)
AGC
VX-680
I
57
107
93
57
107
93
A
2ETKA_HFS
(ROCK1)
AGC
HMS2231N23
I
6
12
24
6
12
24
A
2JDRA_L20
(AKT2)
AGC
A-443654
I
44
255
61
44
255
61
A
2H8HA_H8H
(SRC)
AGC
Saracatinib
I
91
255
126
91
255
126
A
3D9VA_H52
(ROCK1)
AGC
H-1152P
I
7
16
24
7
16
24
A
2IVUA_ZD6
(RET)
AGC
Vandetanib
I
83
291
121
83
291
121
A
3FC2A_IBI
(PLK1)
AGC
BI 2536
I
38
72
42
38
72
42
A
2JEDA_LG8
(PRKCQ)
AGC
5-Arylidene-...
I
67
19
87
67
19
87
A
2IW6A_QQ2
(CDK2)
AGC
2iw6
I
112
209
86
112
209
86
A
3KRWA_BA1
(ADRBK1)
AGC
balanol
I
17
127
29
17
127
29
A
1NVSA_UCM
(CHEK1)
AGC
SB218078
I
97
6
53
97
6
53
A
2F4JA_VX6
(ABL1)
AGC
VX-680
I
110
109
134
110
109
134
A
2I40A_BLZ
(CDK2)
AGC
2i40
I
34
95
16
34
95
16
A
2WIHA_P48
(CDK2)
AGC
VX_680
I
111
425
105
111
425
105
A
3D0EA_G93
(AKT2)
AGC
9-N-ethyl-8-...
I
30
15
45
30
15
45
A
2XYNA_VX6
(ABL2)
AGC
VX-680
I
79
101
105
79
101
105
B
21
3BKBA_STU
(FES)
AGC
staurosporine
I
131
107
138
B
3BKBA_STU
(FES)
AGC
staurosporine
I
131
107
138
131
107
138
B
3CBLA_STU
(FES)
AGC
staurosporine
I
131
107
138
131
107
138
B
1WVYA_STU
(DAPK1)
AGC
staurosporine
I
83
23
55
83
23
55
B
3CD3A_STU
(FES)
AGC
staurosporine
I
131
107
138
131
107
138
B
1OKYA_STU
(PDPK1)
AGC
staurosporine
I
179
67
109
179
67
109
B
1OKZA_UCN
(PDPK1)
AGC
UCN 02
I
179
60
109
179
60
109
B
2PE2A_464
(PDPK1)
AGC
Indolinone b...
I
134
156
104
134
156
104
B
1UVRA_BI8
(PDPK1)
AGC
Ro 31-7549
I
82
181
65
82
181
65
B
1UU3A_LY4
(PDPK1)
AGC
Ruboxistaurin
I
71
117
57
71
117
57
B
1UU7A_BI2
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
3ORZA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU8A_BI1
(PDPK1)
AGC
bisindolylma...
I
83
189
65
83
189
65
B
3OTUA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU9A_BI3
(PDPK1)
AGC
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
3NCZA_3NC
(ROCK1)
AGC
Cis-4-Amino-...
I
4
41
3
4
41
3
B
3NYNA_SGV
(GRK6)
AGC
SMR000127424
I
54
7
47
54
7
47
B
2FVDA_LIA
(CDK2)
AGC
[4-Amino-2-[...
I
39
16
29
39
16
29
B
2ESMA_M77
(ROCK1)
AGC
HMS2231N23
I
6
15
24
6
15
24
B
1H07A_MFP
(CDK2)
AGC
AC1NAKJQ
I
90
241
80
90
241
80
B
2BMCA_MPY
(AURKA)
AGC
PHA-680632
I
107
108
107
107
108
107
B
3KRXA_BA1
(ADRBK1)
AGC
balanol
I
14
106
29
14
106
29