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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
1 PRKCH related diseases
601367
{Cerebral infarction, susceptibility to}
Summary of query kinase
Query kinase
PRKCH (
P24723
)
Kinase group
AGC
Number of conformation types
0
Number of structural templates
42 (
Total 183 inhibitors
)
Number of PRKCH related diseases
1 (
601367
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
30
3KRWA_BA1
(ADRBK1)
AGC
balanol
I
17
127
29
A
3KRWA_BA1
(ADRBK1)
AGC
balanol
I
17
127
29
17
127
29
A
2BILB_BI1
(PIM1)
AGC
bisindolylma...
I
41
132
36
41
132
36
A
2I0EA_PDS
(PRKCB)
AGC
bisindolylma...
I
41
141
45
41
141
45
A
1XWSA_BI1
(PIM1)
AGC
bisindolylma...
I
41
132
36
41
132
36
A
2BIKB_BI1
(PIM1)
AGC
bisindolylma...
I
41
132
36
41
132
36
A
2J2IB_LY4
(PIM1)
AGC
Ruboxistaurin
I
35
89
36
35
89
36
A
3IW4A_LW4
(PRKCA)
AGC
Sotrastaurin
I
52
119
49
52
119
49
A
1NVRA_STU
(CHEK1)
AGC
staurosporine
I
179
71
79
179
71
79
A
1NXKA_STU
(MAPKAPK2)
AGC
staurosporine
I
110
67
51
110
67
51
A
1AQ1A_STU
(CDK2)
AGC
staurosporine
I
195
76
118
195
76
118
A
1XJDA_STU
(PRKCQ)
AGC
staurosporine
I
121
101
106
121
101
106
A
1BYGA_STU
(CSK)
AGC
staurosporine
I
85
72
123
85
72
123
A
1YHSA_STU
(PIM1)
AGC
staurosporine
I
78
64
50
78
64
50
A
1YVJA_4ST
(JAK3)
AGC
staurosporine
I
96
90
126
96
90
126
A
2HZ4A_4ST
(ABL1)
AGC
staurosporine
I
159
103
156
159
103
156
A
1NVQA_UCN
(CHEK1)
AGC
UCN 02
I
179
65
79
179
65
79
A
1PKDA_UCN
(CDK2)
AGC
UCN 02
I
195
67
118
195
67
118
A
2HY81_1ST
(PAK1)
AGC
UCN 02
I
58
20
75
58
20
75
A
3NLBA_5BE
(CHEK1)
AGC
38P
I
45
115
49
45
115
49
A
3A2CA_PDY
(MAPKAPK2)
AGC
6-(4-methoxy...
I
32
39
21
32
39
21
A
1NVSA_UCM
(CHEK1)
AGC
SB218078
I
97
6
53
97
6
53
A
2JEDA_LG8
(PRKCQ)
AGC
5-Arylidene-...
I
67
19
87
67
19
87
A
3D0EA_G93
(AKT2)
AGC
9-N-ethyl-8-...
I
30
15
45
30
15
45
A
2HY0A_306
(CHEK1)
AGC
AMG_706
I
23
80
49
23
80
49
A
2VN9A_GVD
(CAMK2D)
AGC
pyrido[4,3-d...
I
16
75
24
16
75
24
A
3PJCA_PJC
(JAK3)
AGC
3-(1h-Indol-...
I
8
11
25
8
11
25
A
3BHHA_5CP
(CAMK2B)
AGC
DCL001071
I
17
45
22
17
45
22
A
3LM0A_EBD
(STK17B)
AGC
DCL001071
I
20
106
24
20
106
24
A
2IW6A_QQ2
(CDK2)
AGC
2iw6
I
112
209
86
112
209
86
A
2JDRA_L20
(AKT2)
AGC
A-443654
I
44
255
61
44
255
61
B
12
1UU8A_BI1
(PDPK1)
AGC
bisindolylma...
I
83
189
65
B
1UU8A_BI1
(PDPK1)
AGC
bisindolylma...
I
83
189
65
83
189
65
B
1UVRA_BI8
(PDPK1)
AGC
Ro 31-7549
I
82
181
65
82
181
65
B
1ZRZA_BI1
(PRKCI)
AGC
bisindolylma...
I
52
150
47
52
150
47
B
1UU7A_BI2
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU9A_BI3
(PDPK1)
AGC
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
3ORZA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
3OTUA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU3A_LY4
(PDPK1)
AGC
Ruboxistaurin
I
71
117
57
71
117
57
B
1OKYA_STU
(PDPK1)
AGC
staurosporine
I
179
67
109
179
67
109
B
1OKZA_UCN
(PDPK1)
AGC
UCN 02
I
179
60
109
179
60
109
B
2PE2A_464
(PDPK1)
AGC
Indolinone b...
I
134
156
104
134
156
104
B
2XCKA_MH4
(PDPK1)
AGC
MH4
I
46
431
75
46
431
75