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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
1 PRKCZ related diseases
hsa04930
Type II diabetes mellitus
Summary of query kinase
Query kinase
PRKCZ (
Q05513
)
Kinase group
AGC
Number of conformation types
0
Number of structural templates
39 (
Total 50 inhibitors
)
Number of PRKCZ related diseases
1 (
hsa04930
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
17
2I0EA_PDS
(PRKCB)
AGC
bisindolylma...
I
41
141
45
A
2I0EA_PDS
(PRKCB)
AGC
bisindolylma...
I
41
141
45
41
141
45
A
3KRWA_BA1
(ADRBK1)
AGC
balanol
I
17
127
29
17
127
29
A
1ZYSA_199
(CHEK1)
AGC
2,4-Diamino-...
I
31
92
52
31
92
52
A
2HY0A_306
(CHEK1)
AGC
AMG_706
I
23
80
49
23
80
49
A
2HOGA_710
(CHEK1)
AGC
3-(Indol-2-y...
I
33
66
51
33
66
51
A
2HXLA_422
(CHEK1)
AGC
DB07075
I
15
95
36
15
95
36
A
3NLBA_5BE
(CHEK1)
AGC
38P
I
45
115
49
45
115
49
A
3CKXA_STU
(STK24)
AGC
staurosporine
I
176
104
141
176
104
141
A
1BYGA_STU
(CSK)
AGC
staurosporine
I
85
72
123
85
72
123
A
1NVQA_UCN
(CHEK1)
AGC
UCN 02
I
179
65
79
179
65
79
A
1NVRA_STU
(CHEK1)
AGC
staurosporine
I
179
71
79
179
71
79
A
1NXKA_STU
(MAPKAPK2)
AGC
staurosporine
I
110
67
51
110
67
51
A
3R2YA_P4O
(MAPKAPK2)
AGC
2jbo
I
18
130
30
18
130
30
A
2JBOA_P4O
(MAPKAPK2)
AGC
2jbo
I
18
130
30
18
130
30
A
2JBPA_P4O
(MAPKAPK2)
AGC
2jbo
I
18
130
30
18
130
30
A
2C3KA_ABO
(CHEK1)
AGC
ABO
I
15
47
31
15
47
31
A
3KGAA_LX9
(MAPKAPK2)
AGC
LX9
I
14
42
21
14
42
21
B
22
3ORZA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
B
3ORZA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU7A_BI2
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
3OTUA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
1UU8A_BI1
(PDPK1)
AGC
bisindolylma...
I
83
189
65
83
189
65
B
1UU9A_BI3
(PDPK1)
AGC
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
1UVRA_BI8
(PDPK1)
AGC
Ro 31-7549
I
82
181
65
82
181
65
B
1ZRZA_BI1
(PRKCI)
AGC
bisindolylma...
I
52
150
47
52
150
47
B
3KRXA_BA1
(ADRBK1)
AGC
balanol
I
14
106
29
14
106
29
B
1UU3A_LY4
(PDPK1)
AGC
Ruboxistaurin
I
71
117
57
71
117
57
B
3IONA_8H1
(PDPK1)
AGC
8H1
I
16
93
51
16
93
51
B
3IOPA_8I1
(PDPK1)
AGC
8H1
I
16
93
51
16
93
51
B
2PE2A_464
(PDPK1)
AGC
Indolinone b...
I
134
156
104
134
156
104
B
1WVYA_STU
(DAPK1)
AGC
staurosporine
I
83
23
55
83
23
55
B
2BMCA_MPY
(AURKA)
AGC
PHA-680632
I
107
108
107
107
108
107
B
1OKYA_STU
(PDPK1)
AGC
staurosporine
I
179
67
109
179
67
109
B
2XRUA_400
(AURKA)
AGC
VX_680
I
33
152
63
33
152
63
B
1OKZA_UCN
(PDPK1)
AGC
UCN 02
I
179
60
109
179
60
109
B
3FHRA_P4O
(MAPKAPK3)
AGC
2jbo
I
17
110
31
17
110
31
B
1OIRA_HDY
(CDK2)
AGC
AC1O6YZF
I
51
203
64
51
203
64
B
3GOKA_P4O
(MAPKAPK2)
AGC
2jbo
I
20
134
35
20
134
35
B
2W1EA_L0E
(AURKA)
AGC
pyrazole-ben...
I
15
32
45
15
32
45
B
3QD0A_3Q4
(PDPK1)
AGC
(3s,6r)-1-[2...
I
28
114
63
28
114
63