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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
PRKG1 (
Q13976
)
Kinase group
AGC
Number of conformation types
0
Number of structural templates
29 (
Total 29 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
11
1NVQA_UCN
(CHEK1)
AGC
UCN 02
I
179
65
79
A
1NVQA_UCN
(CHEK1)
AGC
UCN 02
I
179
65
79
179
65
79
A
1NVRA_STU
(CHEK1)
AGC
staurosporine
I
179
71
79
179
71
79
A
2HZ4A_4ST
(ABL1)
AGC
staurosporine
I
159
103
156
159
103
156
A
2JDOA_I5S
(AKT2)
AGC
I5S
I
10
22
29
10
22
29
A
1NVSA_UCM
(CHEK1)
AGC
SB218078
I
97
6
53
97
6
53
A
1ZZLA_TZY
(MAPK14)
AGC
CP-808844
I
36
84
44
36
84
44
A
2JDRA_L20
(AKT2)
AGC
A-443654
I
44
255
61
44
255
61
A
3D0EA_G93
(AKT2)
AGC
9-N-ethyl-8-...
I
30
15
45
30
15
45
A
3L8XA_N4D
(MAPK14)
AGC
3cg2
I
91
104
65
91
104
65
A
3HA8A_5JZ
(MAPK14)
AGC
DEL-B, 14b
I
59
89
62
59
89
62
A
1BL6A_SB6
(MAPK14)
AGC
sb216995
I
46
110
50
46
110
50
B
18
1OKYA_STU
(PDPK1)
AGC
staurosporine
I
179
67
109
B
1OKYA_STU
(PDPK1)
AGC
staurosporine
I
179
67
109
179
67
109
B
1OKZA_UCN
(PDPK1)
AGC
UCN 02
I
179
60
109
179
60
109
B
1WVYA_STU
(DAPK1)
AGC
staurosporine
I
83
23
55
83
23
55
B
1UU8A_BI1
(PDPK1)
AGC
bisindolylma...
I
83
189
65
83
189
65
B
1UU9A_BI3
(PDPK1)
AGC
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
1UVRA_BI8
(PDPK1)
AGC
Ro 31-7549
I
82
181
65
82
181
65
B
1MUOA_ADN
(AURKA)
AGC
Vidarabine
I
11
12
32
11
12
32
B
1ZRZA_BI1
(PRKCI)
AGC
bisindolylma...
I
52
150
47
52
150
47
B
3ORZA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
3OTUA_BI4
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
3NYNA_SGV
(GRK6)
AGC
SMR000127424
I
54
7
47
54
7
47
B
1UU7A_BI2
(PDPK1)
AGC
bisindolylma...
I
82
178
65
82
178
65
B
3KRXA_BA1
(ADRBK1)
AGC
balanol
I
14
106
29
14
106
29
B
2VZ6A_FEF
(CAMK2A)
AGC
indirubin de...
I
15
3
14
15
3
14
B
3L9MA_L9M
(PRKACA)
AGC
VX_680
I
37
65
42
37
65
42
B
2BMCA_MPY
(AURKA)
AGC
PHA-680632
I
107
108
107
107
108
107
B
2PE2A_464
(PDPK1)
AGC
Indolinone b...
I
134
156
104
134
156
104
B
1UU3A_LY4
(PDPK1)
AGC
Ruboxistaurin
I
71
117
57
71
117
57