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Example2
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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
G95
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
AKT2 (PDB code: 3E87)
[PDB]
[PDBsum]
Inhibitor
AG_013736 (HET code: G95)
[PDB]
Summary of KIF 3E87A_G95
(AKT2, PDB code:
3E87
, chain A)
Number of family interactions
73
Number of family kinase
9 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
42 (12 are AKT2 inhibitors)
Involved diseases
28 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
AKT2 and 12 inhibitors