Protein Surface  Ribbon
Inhibitor XBJ
  ATP Location
Pocket ATP NLP HAP CLP SP
Selected template
Kinase CHEK2 (PDB code: 2XBJ) [PDB] [PDBsum]
Inhibitor 4-Fluoro-2-(4-{[(3s,4r)-4-(1-Hydroxy-1-Methylethyl)pyrrolidin-3-Yl]amino}-6,7-Dimethoxyquinazolin-2-Yl)phenol (HET code: XBJ) [PDB]
 
Summary of KIF 2XBJA_XBJ (CHEK2, PDB code: 2XBJ, chain A)
Number of family interactions 40
Number of family kinase 2 (sequence conservation) (profiling results)
Number of family inhibitors 24 (24 are CHEK2 inhibitors)
Involved diseases 4 (show)
Number of family anchors  
All kinase-inhibitor interactions in this family  CHEK2 and 24 inhibitors