Protein Surface  Ribbon
Inhibitor DFZ
  ATP Location
Pocket ATP NLP HAP CLP SP
Selected template
Kinase CHEK1 (PDB code: 2BRM) [PDB] [PDBsum]
Inhibitor DFZ (HET code: DFZ) [PDB]
 
Summary of KIF 2BRMA_DFZ (CHEK1, PDB code: 2BRM, chain A)
Number of family interactions 131
Number of family kinase 21 (sequence conservation) (profiling results)
Number of family inhibitors 88 (1 are RPS6KA2 inhibitors)
Involved diseases 36 (show)
Number of family anchors  
All kinase-inhibitor interactions in this family  RPS6KA2 and 1 inhibitors