Protein Surface  Ribbon
Inhibitor S22
  ATP Location
Pocket ATP NLP HAP CLP SP
Selected template
Kinase TTK (PDB code: 3GFW) [PDB] [PDBsum]
Inhibitor 1-(4-(4-(2-(Isopropylsulfonyl)phenylamino)-1H-pyrrolo[2,3-b]pyridin-6-ylamino)-3-methoxyphenyl)piperidin-4-ol (HET code: S22) [PDB]
 
Summary of KIF 3GFWA_S22 (TTK, PDB code: 3GFW, chain A)
Number of family interactions 42
Number of family kinase 21 (sequence conservation) (profiling results)
Number of family inhibitors 4 (2 are RPS6KA2 inhibitors)
Involved diseases 18 (show)
Number of family anchors  
All kinase-inhibitor interactions in this family  RPS6KA2 and 2 inhibitors