Summary of query kinase
Query kinase ACVR2A (P27037)
Kinase group TKL
Number of inhibitors 15
Index Target Inhibitor Inhibitor 2D Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) POC Source Link
0 ACVR2A PD_173955 PD_173955 n/a n/a 10 n/a n/a NB2011DRx NB2011DRx
1 ACVR2A PP_242 PP_242 n/a n/a 18 n/a n/a NB2011DRx NB2011DRx
2 ACVR2A BMS-354825 BD00013216 n/a n/a 210 n/a n/a BindingDB BindingDB
3 ACVR2A Dasatinib Dasatinib n/a n/a 210 n/a n/a NB2008 NB2008
4 ACVR2A Dasatinib Dasatinib n/a n/a 210 n/a n/a NB2011DRx NB2011DRx
5 ACVR2A TAE_684 TAE_684 n/a n/a 2200 n/a n/a NB2011DRx NB2011DRx
6 ACVR2A CHEMBL603469 BD50308060 n/a n/a 2500 n/a n/a BindingDB BindingDB
7 ACVR2A CEP_701 CEP_701 n/a n/a 2500 n/a n/a NB2011DRx NB2011DRx
8 ACVR2A JNJ-7706621 BD00006866 n/a n/a 2900 n/a n/a BindingDB BindingDB
9 ACVR2A JNJ_7706621 JNJ_7706621 n/a n/a 2900 n/a n/a NB2008 NB2008
10 ACVR2A Flavopiridol Flavopiridol n/a n/a 3100 n/a n/a NB2011DRx NB2011DRx
11 ACVR2A KW_2449 KW_2449 n/a n/a 320 n/a n/a NB2011DRx NB2011DRx
12 ACVR2A Staurosporine Staurosporine n/a n/a 8900 n/a n/a NB2011DRx NB2011DRx
13 ACVR2A GVD GVD n/a n/a n/a n/a n/a PDB PDB
14 ACVR2A TAK TAK n/a n/a n/a n/a n/a PDB PDB