Kinase profiling results of kinases in KIF 1OIRA_HDY (CDK2, PDB code: 1OIR, chain A)
Template Kinase: CDK2
Template inhibitor: AC1O6YZF

51 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C C C
AKT1AGC   
AKT2AGC   
PDPK1AGC   
PRKCDAGC   
PRKCQAGC   
PRKCEAGC   
PKN1AGC   
CHEK1CAMK   
STK17ACAMK   
PHKG1CAMK   
PHKG2CAMK   
CDK2CMGC   
CDK4CMGC   
CDK7CMGC   
CDK9CMGC   
CLK1CMGC   
CLK2CMGC   
CLK4CMGC   
DYRK1ACMGC   
DYRK1BCMGC   
DYRK2CMGC   
GSK3BCMGC   
MAPK10CMGC   
AURKAOther   
CAMKK2Other   
PLK1Other   
MAP2K1STE   
ABL1TK   
TNK2TK   
EPHA1TK   
EPHB1TK   
PTK2TK   
JAK3TK   
METTK   
MUSKTK   
FGRTK   
FYNTK   
SRCTK   
YES1TK   
BLKTK   
LCKTK   
PTK6TK   
ZAP70TK   
ITKTK   
NTRK2TK   
NTRK3TK   
MAP3K7TKL   

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C C C
AKT1AGC      
AKT2AGC      
PDPK1AGC      
PKN1AGC      
PRKCAAGC      
PRKCDAGC      
PRKCEAGC      
PRKCQAGC      
PRKCZAGC      
CHEK1CAMK      
PHKG1CAMK      
PHKG2CAMK      
STK17ACAMK      
CDC2CMGC      
CDC2CMGC      
CDK2CMGC      
CDK4CMGC      
CDK6CMGC      
CDK6CMGC      
CDK7CMGC      
CDK9CMGC      
CLK1CMGC      
CLK2CMGC      
CLK4CMGC      
DYRK1ACMGC      
DYRK1BCMGC      
DYRK2CMGC      
GSK3BCMGC      
MAPK10CMGC      
AURKAOther      
CAMKK2Other      
PLK1Other      
MAP2K1STE      
ABL1TK      
BLKTK      
EPHA1TK      
EPHB1TK      
FGRTK      
FYNTK      
ITKTK      
JAK3TK      
LCKTK      
METTK      
MUSKTK      
NTRK2TK      
NTRK3TK      
PTK2TK      
PTK6TK      
SRCTK      
TNK2TK      
YES1TK      
ZAP70TK      
MAP3K7TKL