Kinase profiling results of kinases in KIF 1R78A_FMD (CDK2, PDB code: 1R78, chain A)
Template Kinase: CDK2
Template inhibitor: 4-alkynyl oxindole 7o

127 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C
ROCK1AGC 
ROCK2AGC 
GRK1AGC 
GRK4AGC 
GRK7AGC 
MAST1AGC 
PDPK1AGC 
PRKCQAGC 
PKN1AGC 
PKN2AGC 
RPS6KA4AGC 
RPS6KA4CAMK 
RPS6KA5AGC 
RPS6KA5CAMK 
RPS6KB1AGC 
RPS6KA1AGC 
RPS6KA1CAMK 
RPS6KA2AGC 
RPS6KA2CAMK 
RPS6KA3AGC 
RPS6KA6AGC 
RPS6KA6CAMK 
SGK3AGC 
CAMK1GCAMK 
CAMK2ACAMK 
CAMK2BCAMK 
CAMK2DCAMK 
BRSK1CAMK 
BRSK2CAMK 
CHEK1CAMK 
HUNKCAMK 
MARK1CAMK 
MARK2CAMK 
MARK3CAMK 
MARK4CAMK 
MGC421053 
NUAK1CAMK 
NUAK2CAMK 
SIK1CAMK 
SIK2CAMK 
SNRKCAMK 
STK33CAMK 
DAPK1CAMK 
DAPK2CAMK 
DAPK3CAMK 
STK17ACAMK 
STK17BCAMK 
PHKG1CAMK 
PHKG2CAMK 
PIM3CAMK 
PRKD1CAMK 
PRKD2CAMK 
PRKD3CAMK 
CHEK2CAMK 
CDK2CMGC 
CDK4CMGC 
PCTK1CMGC 
PCTK3CMGC 
PFTK1CMGC 
CDKL2CMGC 
CSNK2A1CMGC 
CSNK2A2CMGC 
CLK1CMGC 
CLK2CMGC 
CLK4CMGC 
DYRK1ACMGC 
DYRK1BCMGC 
DYRK2CMGC 
HIPK1CMGC 
HIPK2CMGC 
HIPK3CMGC 
HIPK4CMGC 
PRPF4BCMGC 
MAPK10CMGC 
MAPK9CMGC 
ICKCMGC 
AURKBOther 
AURKCOther 
CAMKK1Other 
CAMKK2Other 
CHUKOther 
NEK2Other 
SBK1Other 
STK35Other 
EIF2AK2Other 
TLK2Other 
TTKOther 
ULK3Other 
PAK3STE 
SLKSTE 
STK10STE 
STK24STE 
STK25STE 
MAP2K1STE 
MAP2K3STE 
MAP2K6STE 
MAP2K5STE 
ABL1TK 
TNK2TK 
AXLTK 
MATKTK 
DDR2TK 
EPHB1TK 
FERTK 
FGFR1TK 
FGFR2TK 
FGFR3TK 
FGFR4TK 
JAK1TK 
JAK2TK 
JAK3TK 
METTK 
MUSKTK 
FRKTK 
FGRTK 
FYNTK 
SRCTK 
YES1TK 
BLKTK 
HCKTK 
LCKTK 
LYNTK 
SRMSTK 
ITKTK 
NTRK2TK 
NTRK3TK 
IRAK4TKL 
MAP3K12TKL 
MAP3K13TKL 
MAP3K11TKL 
MAP3K9TKL 
MAP3K7TKL 

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group
GRK4AGC
GRK7AGC
PDPK1AGC
PKN1AGC
PKN2AGC
PRKCQAGC
ROCK1AGC
ROCK2AGC
RPS6KA1AGC
RPS6KA2AGC
RPS6KA3AGC
RPS6KA4AGC
RPS6KA5AGC
RPS6KA6AGC
RPS6KB1AGC
SGK3AGC
BRSK1CAMK
BRSK2CAMK
CAMK1GCAMK
CAMK2ACAMK
CAMK2BCAMK
CAMK2DCAMK
CHEK1CAMK
CHEK2CAMK
DAPK1CAMK
DAPK2CAMK
DAPK3CAMK
MARK1CAMK
MARK2CAMK
MARK3CAMK
MARK4CAMK
NUAK1CAMK
NUAK2CAMK
PHKG1CAMK
PHKG2CAMK
PIM3CAMK
PRKD1CAMK
PRKD2CAMK
PRKD3CAMK
SIK2CAMK
STK17ACAMK
STK33CAMK
CDK2CMGC
CDK4CMGC
CLK1CMGC
CLK2CMGC
CLK4CMGC
CSNK2A1CMGC
CSNK2A2CMGC
DYRK1ACMGC
DYRK1BCMGC
DYRK2CMGC
HIPK1CMGC
HIPK2CMGC
HIPK3CMGC
HIPK4CMGC
MAPK10CMGC
MAPK9CMGC
AURKBOther
AURKCOther
CAMKK1Other
CAMKK2Other
CHUKOther
NEK2Other
TLK2Other
TTKOther
ULK3Other
MAP2K1STE
MAP2K6STE
PAK3STE
SLKSTE
STK10STE
STK24STE
STK25STE
ABL1TK
AXLTK
BLKTK
DDR2TK
EPHB1TK
FERTK
FGFR1TK
FGFR2TK
FGFR3TK
FGFR4TK
FGRTK
FRKTK
FYNTK
HCKTK
ITKTK
JAK1TK
JAK2TK
JAK3TK
LCKTK
LYNTK
MATKTK
METTK
MUSKTK
NTRK2TK
NTRK3TK
SRCTK
SRMSTK
TNK2TK
YES1TK
IRAK4TKL
MAP3K11TKL
MAP3K7TKL
MAP3K9TKL