Kinase profiling results of kinases in KIF 2BHEA_BRY (CDK2, PDB code: 2BHE, chain A)
Template Kinase: CDK2
Template inhibitor: BRY

51 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group
PDPK1AGC
RPS6KA1AGC
RPS6KA1CAMK
RPS6KA2AGC
RPS6KA2CAMK
RPS6KA6AGC
RPS6KA6CAMK
CAMK2ACAMK
CAMK2DCAMK
BRSK1CAMK
BRSK2CAMK
NUAK1CAMK
SIK2CAMK
STK17ACAMK
PHKG1CAMK
PIM1CAMK
PIM2CAMK
PIM3CAMK
CHEK2CAMK
CDK2CMGC
CDK3CMGC
CDK5CMGC
CDK9CMGC
CSNK2A1CMGC
CSNK2A2CMGC
DYRK1ACMGC
GSK3ACMGC
GSK3BCMGC
NLKCMGC
AURKAOther
AURKBOther
AURKCOther
EIF2AK2Other
ABL1TK
ABL2TK
TNK2TK
FGFR1TK
FRKTK
FGRTK
FYNTK
SRCTK
YES1TK
BLKTK
HCKTK
LCKTK
LYNTK
BMXTK
ITKTK
NTRK2TK
NTRK3TK
MAP3K11TKL
MAP3K9TKL

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C
PDPK1AGC    
RPS6KA1AGC    
RPS6KA2AGC    
RPS6KA6AGC    
BRSK1CAMK    
BRSK2CAMK    
CAMK2ACAMK    
CAMK2DCAMK    
CHEK2CAMK    
NUAK1CAMK    
PHKG1CAMK    
PIM1CAMK    
PIM2CAMK    
PIM3CAMK    
SIK2CAMK    
STK17ACAMK    
CDC2CMGC    
CDC2CMGC    
CDK2CMGC    
CDK3CMGC    
CDK5CMGC    
CDK6CMGC    
CDK6CMGC    
CDK9CMGC    
CSNK2A1CMGC    
CSNK2A2CMGC    
DYRK1ACMGC    
GSK3ACMGC    
GSK3BCMGC    
NLKCMGC    
AURKAOther    
AURKBOther    
AURKCOther    
ABL1TK    
ABL2TK    
BLKTK    
BMXTK    
FGFR1TK    
FGRTK    
FRKTK    
FYNTK    
HCKTK    
ITKTK    
LCKTK    
LYNTK    
NTRK2TK    
NTRK3TK    
SRCTK    
TNK2TK    
YES1TK    
MAP3K11TKL    
MAP3K9TKL