Kinase profiling results of kinases in KIF 2R3NA_SCZ (CDK2, PDB code: 2R3N, chain A)
Template Kinase: CDK2
Template inhibitor: AC1LZZHM

46 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C C
AKT1AGC  
ROCK1AGC  
ROCK2AGC  
PDPK1AGC  
PRKCDAGC  
PRKCQAGC  
CHEK1CAMK  
NUAK1CAMK  
STK33CAMK  
DAPK1CAMK  
PIM1CAMK  
CHEK2CAMK  
CDK2CMGC  
CDK4CMGC  
CSNK2A1CMGC  
CSNK2A2CMGC  
CLK3CMGC  
CLK4CMGC  
GSK3ACMGC  
GSK3BCMGC  
MAPK10CMGC  
MAPK14CMGC  
AURKAOther  
AURKBOther  
CHUKOther  
EIF2AK2Other  
PLK1Other  
SLKSTE  
ABL1TK  
ABL2TK  
TNK2TK  
FERTK  
FGFR1TK  
JAK2TK  
JAK3TK  
FYNTK  
SRCTK  
YES1TK  
LCKTK  
BMXTK  
ITKTK  
NTRK2TK  
NTRK3TK  
MAP3K11TKL  
MAP3K9TKL  

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C
AKT1AGC    
PDPK1AGC    
PRKCDAGC    
PRKCQAGC    
ROCK1AGC    
ROCK2AGC    
CHEK1CAMK    
CHEK2CAMK    
DAPK1CAMK    
NUAK1CAMK    
PIM1CAMK    
STK33CAMK    
CDC2CMGC    
CDC2CMGC    
CDK2CMGC    
CDK4CMGC    
CLK3CMGC    
CLK4CMGC    
CSNK2A1CMGC    
CSNK2A2CMGC    
GSK3ACMGC    
GSK3BCMGC    
MAPK10CMGC    
MAPK14CMGC    
AURKAOther    
AURKBOther    
CHUKOther    
PLK1Other    
SLKSTE    
ABL1TK    
ABL2TK    
BMXTK    
FERTK    
FGFR1TK    
FYNTK    
ITKTK    
JAK2TK    
JAK3TK    
LCKTK    
NTRK2TK    
NTRK3TK    
SRCTK    
TNK2TK    
YES1TK    
MAP3K11TKL    
MAP3K9TKL