Kinase profiling results of kinases in KIF 3NS9A_NS9 (CDK2, PDB code: 3NS9, chain A)
Template Kinase: CDK2
Template inhibitor: pyrazolo[1,5-a]-1,3,5-triazine, 7b

44 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group
ROCK2AGC
CHEK1CAMK
DAPK1CAMK
CHEK2CAMK
CDK2CMGC
CDK3CMGC
CDK4CMGC
CDK5CMGC
CDK7CMGC
CDK9CMGC
PCTK1CMGC
CLK1CMGC
CLK2CMGC
CLK4CMGC
DYRK1ACMGC
DYRK1BCMGC
GSK3BCMGC
MAPK1CMGC
MAPK3CMGC
MAPK15CMGC
AURKAOther
CAMKK2Other
CHUKOther
PLK1Other
PLK3Other
TTKOther
PAK4STE
PAK7STE
SLKSTE
ABL1TK
TNK2TK
JAK2TK
JAK3TK
MUSKTK
FGRTK
FYNTK
SRCTK
YES1TK
HCKTK
ZAP70TK
NTRK2TK
NTRK3TK

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C C C
ROCK2AGC      
CHEK1CAMK      
CHEK2CAMK      
DAPK1CAMK      
CDC2CMGC      
CDC2CMGC      
CDK2CMGC      
CDK3CMGC      
CDK4CMGC      
CDK5CMGC      
CDK6CMGC      
CDK6CMGC      
CDK7CMGC      
CDK9CMGC      
CLK1CMGC      
CLK2CMGC      
CLK4CMGC      
DYRK1ACMGC      
DYRK1BCMGC      
GSK3BCMGC      
MAPK1CMGC      
MAPK3CMGC      
AURKAOther      
CAMKK2Other      
CHUKOther      
PLK1Other      
PLK3Other      
TTKOther      
PAK4STE      
PAK7STE      
SLKSTE      
ABL1TK      
FGRTK      
FYNTK      
HCKTK      
JAK2TK      
JAK3TK      
MUSKTK      
NTRK2TK      
NTRK3TK      
SRCTK      
TNK2TK      
YES1TK      
ZAP70TK