BioXGEM.
KIDFamMap
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Example1
Example2
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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
14 ERBB2 related diseases
H00018
Gastric cancer
H00019
Pancreatic cancer
H00022
Bladder cancer
H00026
Endometrial Cancer
H00027
Ovarian cancer
H00028
Choriocarcinoma
H00030
Cervical cancer
H00031
Breast cancer
H00046
Cholangiocarcinoma
hsa05215
Prostate cancer
211980
Adenocarcinoma of lung, somatic
137215
Gastric cancer, somatic
137800
Glioblastoma, somatic
OMIM
(164870)
Ovarian cancer, somatic,
Summary of query kinase
Query kinase
ERBB2 (
P04626
)
Kinase group
TK
Number of conformation types
1
Number of structural templates
1 (
Total 935 inhibitors
)
Number of ERBB2 related diseases
14 (
H00018
H00019
H00022
H00026
H00027
H00028
H00030
H00031
...
)
Number of allelic variants
6 (
E914K
G776S
L755P
N857S
V654I
V655I
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
1
3PP0A_03Q
(ERBB2)
TK
AZD_1152HQPA
I
3
21
20
A
3PP0A_03Q
(ERBB2)
TK
AZD_1152HQPA
I
3
21
20
3
21
20