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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
2 PAK3 related diseases
H00480
Non-syndromic X-linked mental retardation
300558
Mental retardation, X-linked 30/47
Summary of query kinase
Query kinase
PAK3 (
O75914
)
Kinase group
STE
Number of conformation types
0
Number of structural templates
38 (
Total 43 inhibitors
)
Number of PAK3 related diseases
2 (
H00480
300558
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
24
1Q3DA_STU
(GSK3B)
STE
staurosporine
I
115
71
61
A
1Q3DA_STU
(GSK3B)
STE
staurosporine
I
115
71
61
115
71
61
A
3CKXA_STU
(STK24)
STE
staurosporine
I
176
104
141
176
104
141
A
1AQ1A_STU
(CDK2)
STE
staurosporine
I
195
76
118
195
76
118
A
1SM2A_STU
(ITK)
STE
staurosporine
I
99
104
128
99
104
128
A
1NVQA_UCN
(CHEK1)
STE
UCN 02
I
179
65
79
179
65
79
A
1SNUA_STU
(ITK)
STE
staurosporine
I
99
104
128
99
104
128
A
1NVRA_STU
(CHEK1)
STE
staurosporine
I
179
71
79
179
71
79
A
1YHSA_STU
(PIM1)
STE
staurosporine
I
78
64
50
78
64
50
A
1NXKA_STU
(MAPKAPK2)
STE
staurosporine
I
110
67
51
110
67
51
A
1PKDA_UCN
(CDK2)
STE
UCN 02
I
195
67
118
195
67
118
A
2HY81_1ST
(PAK1)
STE
UCN 02
I
58
20
75
58
20
75
A
2WIHA_P48
(CDK2)
STE
VX_680
I
111
425
105
111
425
105
A
1R78A_FMD
(CDK2)
STE
4-alkynyl ox...
I
127
24
97
127
24
97
A
2VTTA_LZD
(CDK2)
STE
pyrazole dia...
I
158
42
111
158
42
111
A
3M2WA_L8I
(MAPKAPK2)
STE
Sunitinib
I
84
90
47
84
90
47
A
2IW6A_QQ2
(CDK2)
STE
2iw6
I
112
209
86
112
209
86
A
2BILB_BI1
(PIM1)
STE
bisindolylma...
I
41
132
36
41
132
36
A
2I0EA_PDS
(PRKCB)
STE
bisindolylma...
I
41
141
45
41
141
45
A
2OW3A_BIM
(GSK3B)
STE
LY_333531
I
62
139
51
62
139
51
A
3IKAA_0UN
(EGFR)
STE
2jkk
I
76
120
108
76
120
108
A
1AGWA_SU2
(FGFR1)
STE
SU 4984
I
77
81
111
77
81
111
A
1XWSA_BI1
(PIM1)
STE
bisindolylma...
I
41
132
36
41
132
36
A
1NVSA_UCM
(CHEK1)
STE
SB218078
I
97
6
53
97
6
53
A
2BIKB_BI1
(PIM1)
STE
bisindolylma...
I
41
132
36
41
132
36
B
14
1OKYA_STU
(PDPK1)
STE
staurosporine
I
179
67
109
B
1OKYA_STU
(PDPK1)
STE
staurosporine
I
179
67
109
179
67
109
B
3BKBA_STU
(FES)
STE
staurosporine
I
131
107
138
131
107
138
B
1OKZA_UCN
(PDPK1)
STE
UCN 02
I
179
60
109
179
60
109
B
3CBLA_STU
(FES)
STE
staurosporine
I
131
107
138
131
107
138
B
3CD3A_STU
(FES)
STE
staurosporine
I
131
107
138
131
107
138
B
3MIYA_B49
(ITK)
STE
Sunitinib
I
70
74
110
70
74
110
B
2PE2A_464
(PDPK1)
STE
Indolinone b...
I
134
156
104
134
156
104
B
1H07A_MFP
(CDK2)
STE
AC1NAKJQ
I
90
241
80
90
241
80
B
1UU7A_BI2
(PDPK1)
STE
bisindolylma...
I
82
178
65
82
178
65
B
1UU8A_BI1
(PDPK1)
STE
bisindolylma...
I
83
189
65
83
189
65
B
3ORZA_BI4
(PDPK1)
STE
bisindolylma...
I
82
178
65
82
178
65
B
1UU9A_BI3
(PDPK1)
STE
3-[1-(3-AMIN...
I
83
180
69
83
180
69
B
3OTUA_BI4
(PDPK1)
STE
bisindolylma...
I
82
178
65
82
178
65
B
1UVRA_BI8
(PDPK1)
STE
Ro 31-7549
I
82
181
65
82
181
65