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KIDFamMap
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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
B49
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
KIT (PDB code: 3G0F)
[PDB]
[PDBsum]
Inhibitor
Sunitinib (HET code: B49)
[PDB]
Summary of KIF 3G0FA_B49
(KIT, PDB code:
3G0F
, chain A)
Number of family interactions
403
Number of family kinase
37 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
40 (7 are FLT4 inhibitors)
Involved diseases
78 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
FLT4 and 7 inhibitors