Kinase profiling results of kinases in KIF 3A4OX_STU (LYN, PDB code: 3A4O, chain X)
Template Kinase: LYN
Template inhibitor: staurosporine

73 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C C
PDPK1AGC  
PRKCEAGC  
PKN1AGC  
BRSK1CAMK  
BRSK2CAMK  
CHEK1CAMK  
MARK2CAMK  
MARK4CAMK  
MGC421053  
NUAK1CAMK  
NUAK2CAMK  
KIAA0999CAMK  
SIK1CAMK  
SIK2CAMK  
SNRKCAMK  
DAPK1CAMK  
DAPK2CAMK  
STK17ACAMK  
STK17BCAMK  
PRKD1CAMK  
PRKD2CAMK  
PRKD3CAMK  
CDK2CMGC  
CDK3CMGC  
CDK5CMGC  
CDC2L5CMGC  
CDKL2CMGC  
CDKL3CMGC  
MAPK14CMGC  
ICKCMGC  
MAKCMGC  
SBK1Other  
ABL1TK  
ABL2TK  
TNK1TK  
TNK2TK  
CSKTK  
MATKTK  
EGFRTK  
EPHA8TK  
EPHB1TK  
EPHB2TK  
EPHB4TK  
EPHB6TK  
PTK2TK  
FGFR1TK  
FGFR2TK  
FGFR3TK  
FGFR4TK  
JAK2TK  
CSF1RTK  
KITTK  
PDGFRATK  
PDGFRBTK  
FRKTK  
FGRTK  
FYNTK  
SRCTK  
YES1TK  
BLKTK  
HCKTK  
LCKTK  
LYNTK  
PTK6TK  
SRMSTK  
SYKTK  
ZAP70TK  
BMXTK  
BTKTK  
ACVR1TKL  

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C
PDPK1AGC    
PKN1AGC    
PRKCAAGC    
PRKCEAGC    
BRSK1CAMK    
BRSK2CAMK    
CHEK1CAMK    
DAPK1CAMK    
DAPK2CAMK    
MARK2CAMK    
MARK4CAMK    
NUAK1CAMK    
NUAK2CAMK    
PRKD1CAMK    
PRKD2CAMK    
PRKD3CAMK    
SIK2CAMK    
STK17ACAMK    
TSSK2CAMK    
CDC2CMGC    
CDC2CMGC    
CDK2CMGC    
CDK3CMGC    
CDK5CMGC    
MAPK14CMGC    
ABL1TK    
ABL2TK    
BLKTK    
BMXTK    
BTKTK    
CSF1RTK    
CSKTK    
EGFRTK    
EPHA8TK    
EPHB1TK    
EPHB2TK    
EPHB4TK    
FGFR1TK    
FGFR2TK    
FGFR3TK    
FGFR4TK    
FGRTK    
FRKTK    
FYNTK    
HCKTK    
JAK2TK    
KITTK    
LCKTK    
LYNTK    
MATKTK    
PDGFRATK    
PDGFRBTK    
PTK2TK    
PTK6TK    
SRCTK    
SRMSTK    
SYKTK    
TNK2TK    
YES1TK    
ZAP70TK    
ACVR1TKL