Kinase profiling results of kinases in KIF 1NVSA_UCM (CHEK1, PDB code: 1NVS, chain A)
Template Kinase: CHEK1
Template inhibitor: SB218078

96 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group
AKT2AGC
AKT3AGC
STK38AGC
PDPK1AGC
PRKACAAGC
PRKXAGC
PRKCDAGC
PRKCQAGC
PRKCEAGC
PRKCHAGC
PRKG1AGC
PRKG2AGC
PKN1AGC
PKN2AGC
RPS6KA4AGC
RPS6KA4CAMK
RPS6KA5AGC
RPS6KA5CAMK
RPS6KB1AGC
RPS6KA1AGC
RPS6KA1CAMK
RPS6KA2AGC
RPS6KA2CAMK
RPS6KA3AGC
RPS6KA6AGC
RPS6KA6CAMK
CAMK2ACAMK
CAMK2BCAMK
CAMK2DCAMK
CAMK2GCAMK
BRSK1CAMK
BRSK2CAMK
CHEK1CAMK
MARK1CAMK
MARK2CAMK
MARK3CAMK
MARK4CAMK
NUAK1CAMK
SIK2CAMK
STK33CAMK
DAPK1CAMK
DAPK2CAMK
DAPK3CAMK
STK17ACAMK
MAPKAPK23
MKNK2CAMK
PHKG1CAMK
PIM1CAMK
PIM2CAMK
PIM3CAMK
PRKD1CAMK
PRKD2CAMK
PRKD3CAMK
CHEK2CAMK
TSSK1BCAMK
CDK2CMGC
CDK4CMGC
CDK5CMGC
CDK9CMGC
CSNK2A1CMGC
CSNK2A2CMGC
GSK3ACMGC
GSK3BCMGC
AURKAOther
AURKBOther
AURKCOther
CAMKK1Other
CAMKK2Other
IKBKEOther
TBK1Other
NEK4Other
TLK2Other
ULK3Other
MAP3K2STE
MAP3K3STE
PAK1STE
PAK2STE
PAK3STE
SLKSTE
STK10STE
STK24STE
STK25STE
JAK1TK
BLKTK
HCKTK
LYNTK
NTRK1TK
NTRK2TK
NTRK3TK
IRAK4TKL
LIMK1TKL

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C
AKT2AGC    
AKT3AGC    
PDPK1AGC    
PKN1AGC    
PKN2AGC    
PRKACAAGC    
PRKACGAGC    
PRKCAAGC    
PRKCBAGC    
PRKCBAGC    
PRKCDAGC    
PRKCEAGC    
PRKCHAGC    
PRKCQAGC    
PRKG1AGC    
PRKG2AGC    
PRKXAGC    
RPS6KA1AGC    
RPS6KA2AGC    
RPS6KA3AGC    
RPS6KA4AGC    
RPS6KA5AGC    
RPS6KA6AGC    
RPS6KB1AGC    
RPS6KB2AGC    
SGK1AGC    
SGK2AGC    
STK38AGC    
BRSK1CAMK    
BRSK2CAMK    
CAMK2ACAMK    
CAMK2BCAMK    
CAMK2DCAMK    
CAMK2GCAMK    
CHEK1CAMK    
CHEK2CAMK    
DAPK1CAMK    
DAPK2CAMK    
DAPK3CAMK    
MAPKAPK2CAMK    
MARK1CAMK    
MARK2CAMK    
MARK3CAMK    
MARK4CAMK    
MKNK2CAMK    
NUAK1CAMK    
PASKCAMK    
PHKG1CAMK    
PIM1CAMK    
PIM2CAMK    
PIM3CAMK    
PRKD1CAMK    
PRKD2CAMK    
PRKD3CAMK    
SIK2CAMK    
STK17ACAMK    
STK33CAMK    
TSSK1BCAMK    
CDC2CMGC    
CDC2CMGC    
CDK2CMGC    
CDK4CMGC    
CDK5CMGC    
CDK6CMGC    
CDK6CMGC    
CDK9CMGC    
CSNK2A1CMGC    
CSNK2A2CMGC    
GSK3ACMGC    
GSK3BCMGC    
AURKAOther    
AURKBOther    
AURKCOther    
CAMKK1Other    
CAMKK2Other    
IKBKEOther    
NEK4Other    
NEK8Other    
TBK1Other    
TLK2Other    
ULK3Other    
MAP3K2STE    
MAP3K3STE    
PAK1STE    
PAK2STE    
PAK3STE    
SLKSTE    
STK10STE    
STK24STE    
STK25STE    
BLKTK    
HCKTK    
JAK1TK    
LYNTK    
NTRK1TK    
NTRK2TK    
NTRK3TK    
IRAK4TKL    
LIMK1TKL