Kinase profiling results of kinases in KIF 2W4OA_DKI (CAMK4, PDB code: 2W4O, chain A)
Template Kinase: CAMK4
Template inhibitor: 5-AMINO-3-{[4-(AMINOSULFONYL)PHENYL]AMINO}-N-(2,6-DIFLUOROPHENYL)-1H-1,2,4-TRIAZOLE-1-CARBOTHIOAMIDE

15 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group
ROCK1AGC
ROCK2AGC
CAMK4CAMK
CAMK2ACAMK
DCLK3CAMK
CDK2CMGC
CDK3CMGC
CDK4CMGC
CDK11ACMGC
CDK11ACMGC
MAPK8CMGC
PAK4STE
PAK7STE
SLKSTE
STK24STE

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C
ROCK1AGC  
ROCK2AGC  
CAMK2ACAMK  
CAMK4CAMK  
CDC2CMGC  
CDC2CMGC  
CDK2CMGC  
CDK3CMGC  
CDK4CMGC  
MAPK8CMGC  
PAK4STE  
PAK7STE  
SLKSTE  
STK24STE