Kinase profiling results of kinases in KIF 1OGUA_ST8 (CDK2, PDB code: 1OGU, chain A)
Template Kinase: CDK2
Template inhibitor: ST8

31 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group
ROCK2AGC
RPS6KA2AGC
RPS6KA2CAMK
RPS6KA3AGC
RPS6KA6AGC
RPS6KA6CAMK
NUAK1CAMK
NUAK2CAMK
TSSK1BCAMK
CDK2CMGC
CDK4CMGC
CLK2CMGC
CLK4CMGC
MAPK14CMGC
AURKAOther
AURKBOther
AURKCOther
EIF2AK2Other
TTKOther
TNK2TK
FERTK
JAK2TK
JAK3TK
YES1TK
LCKTK
PTK6TK
BMXTK
NTRK3TK
MAP3K10TKL
MAP3K11TKL
MAP3K9TKL

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C
ROCK2AGC  
RPS6KA2AGC  
RPS6KA3AGC  
RPS6KA6AGC  
NUAK1CAMK  
NUAK2CAMK  
TSSK1BCAMK  
CDC2CMGC  
CDC2CMGC  
CDK2CMGC  
CDK4CMGC  
CDK6CMGC  
CDK6CMGC  
CLK2CMGC  
CLK4CMGC  
MAPK14CMGC  
AURKAOther  
AURKBOther  
AURKCOther  
TTKOther  
BMXTK  
FERTK  
JAK2TK  
JAK3TK  
LCKTK  
NTRK3TK  
PTK6TK  
TNK2TK  
YES1TK  
MAP3K10TKL  
MAP3K11TKL  
MAP3K9TKL