Kinase profiling results of kinases in KIF 1WVYA_STU (DAPK1, PDB code: 1WVY, chain A)
Template Kinase: DAPK1
Template inhibitor: staurosporine

83 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C C
GRK1AGC  
GRK4AGC  
GRK7AGC  
PDPK1AGC  
PRKACAAGC  
PRKACBAGC  
PRKXAGC  
PRKCDAGC  
PRKCQAGC  
PRKCIAGC  
PRKG1AGC  
PRKG2AGC  
PKN2AGC  
RPS6KB1AGC  
CAMK1GCAMK  
CAMK4CAMK  
CAMK2ACAMK  
CHEK1CAMK  
STK33CAMK  
DAPK1CAMK  
DAPK2CAMK  
DAPK3CAMK  
DCLK3CAMK  
MAPKAPK23  
PIM1CAMK  
PIM3CAMK  
PRKD1CAMK  
PRKD2CAMK  
PRKD3CAMK  
CHEK2CAMK  
CDK2CMGC  
CDK3CMGC  
CDK4CMGC  
CDC2L6CMGC  
CDK8CMGC  
CDK9CMGC  
CDKL1CMGC  
CDKL2CMGC  
CSNK2A1CMGC  
HIPK1CMGC  
HIPK2CMGC  
HIPK3CMGC  
HIPK4CMGC  
MAPK1CMGC  
MAPK10CMGC  
MAPK8CMGC  
NLKCMGC  
MAPK12CMGC  
MAPK14CMGC  
ICKCMGC  
MAKCMGC  
AURKAOther  
AURKBOther  
AURKCOther  
TBK1Other  
SBK1Other  
EIF2AK2Other  
TLK2Other  
STK36Other  
ULK3Other  
SLKSTE  
STK24STE  
STK25STE  
ABL1TK  
EPHB1TK  
EPHB2TK  
EPHB4TK  
FERTK  
FESTK  
JAK1TK  
JAK2TK  
BLKTK  
HCKTK  
ZAP70TK  
BMXTK  
BTKTK  

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C
GRK4AGC    
GRK5AGC    
GRK6AGC    
GRK7AGC    
PDPK1AGC    
PKN2AGC    
PRKACAAGC    
PRKACGAGC    
PRKCDAGC    
PRKCIAGC    
PRKCQAGC    
PRKCZAGC    
PRKG1AGC    
PRKG2AGC    
PRKXAGC    
RPS6KB1AGC    
RPS6KB2AGC    
CAMK1GCAMK    
CAMK2ACAMK    
CAMK4CAMK    
CHEK1CAMK    
CHEK2CAMK    
DAPK1CAMK    
DAPK2CAMK    
DAPK3CAMK    
MAPKAPK2CAMK    
PIM1CAMK    
PIM3CAMK    
PRKD1CAMK    
PRKD2CAMK    
PRKD3CAMK    
STK33CAMK    
CDC2CMGC    
CDC2CMGC    
CDK2CMGC    
CDK3CMGC    
CDK4CMGC    
CDK6CMGC    
CDK6CMGC    
CDK9CMGC    
CSNK2A1CMGC    
HIPK1CMGC    
HIPK2CMGC    
HIPK3CMGC    
HIPK4CMGC    
MAPK1CMGC    
MAPK10CMGC    
MAPK12CMGC    
MAPK14CMGC    
MAPK8CMGC    
NLKCMGC    
AURKAOther    
AURKBOther    
AURKCOther    
TBK1Other    
TLK2Other    
ULK3Other    
SLKSTE    
STK24STE    
STK25STE    
ABL1TK    
BLKTK    
BMXTK    
BTKTK    
EPHB1TK    
EPHB2TK    
EPHB4TK    
FERTK    
FESTK    
HCKTK    
JAK1TK    
JAK2TK    
ZAP70TK