Kinase profiling results of kinases in KIF 1XBBA_STI (SYK, PDB code: 1XBB, chain A)
Template Kinase: SYK
Template inhibitor: Imatinib

31 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C C C C C C C
STK17ACAMK       
ABL1TK       
ABL2TK       
ALKTK       
DDR1TK       
EGFRTK       
ERBB4TK       
EPHA8TK       
FGFR1TK       
INSRTK       
JAK2TK       
JAK3TK       
TYK2TK       
CSF1RTK       
KITTK       
PDGFRATK       
PDGFRBTK       
RETTK       
FRKTK       
FGRTK       
FYNTK       
SRCTK       
YES1TK       
BLKTK       
HCKTK       
LCKTK       
LYNTK       
SYKTK       
ITKTK       
BRAFTKL       

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C C C
PRKCAAGC      
STK17ACAMK      
ABL1TK      
ABL2TK      
ALKTK      
BLKTK      
CSF1RTK      
EGFRTK      
EPHA8TK      
ERBB4TK      
FGFR1TK      
FGRTK      
FRKTK      
FYNTK      
HCKTK      
INSRTK      
ITKTK      
JAK2TK      
JAK3TK      
KITTK      
LCKTK      
LYNTK      
PDGFRATK      
PDGFRBTK      
RETTK      
SRCTK      
SYKTK      
TYK2TK      
YES1TK      
BRAFTKL