Kinase profiling results of kinases in KIF 2VWUA_7X1 (EPHB4, PDB code: 2VWU, chain A)
Template Kinase: EPHB4
Template inhibitor: Chlorobenzodioxole deriv. 28

77 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C C C C C C C C
PRKD1CAMK        
PRKD2CAMK        
PRKD3CAMK        
AURKCOther        
NEK4Other        
YSK4STE        
STK39STE        
STK24STE        
ABL1TK        
ABL2TK        
TNK2TK        
ALKTK        
LTKTK        
CSKTK        
MATKTK        
DDR1TK        
DDR2TK        
EGFRTK        
ERBB3TK        
ERBB4TK        
EPHA1TK        
EPHA2TK        
EPHA3TK        
EPHA4TK        
EPHA5TK        
EPHA6TK        
EPHA8TK        
EPHB1TK        
EPHB2TK        
EPHB3TK        
EPHB4TK        
EPHB6TK        
PTK2BTK        
FERTK        
FESTK        
FGFR1TK        
FGFR2TK        
FGFR3TK        
FGFR4TK        
IGF1RTK        
INSRTK        
INSRRTK        
JAK2TK        
TYK2TK        
CSF1RTK        
RETTK        
FRKTK        
FGRTK        
FYNTK        
SRCTK        
YES1TK        
BLKTK        
HCKTK        
LCKTK        
LYNTK        
PTK6TK        
SRMSTK        
SYKTK        
ZAP70TK        
BMXTK        
BTKTK        
ITKTK        
TECTK        
TXKTK        
TEKTK        
TIE1TK        
NTRK1TK        
NTRK2TK        
NTRK3TK        
FLT4TK        
KDRTK        
IRAK1TKL        
IRAK3TKL        
IRAK4TKL        
ACVR1TKL        
ACVR1BTKL        
TGFBR1TKL        

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C
PRKD1CAMK    
PRKD2CAMK    
PRKD3CAMK    
AURKCOther    
NEK4Other    
STK24STE    
STK39STE    
ABL1TK    
ABL2TK    
ALKTK    
BLKTK    
BMXTK    
BTKTK    
CSF1RTK    
CSKTK    
DDR2TK    
EGFRTK    
EPHA1TK    
EPHA2TK    
EPHA3TK    
EPHA4TK    
EPHA5TK    
EPHA6TK    
EPHA8TK    
EPHB1TK    
EPHB2TK    
EPHB3TK    
EPHB4TK    
ERBB4TK    
FERTK    
FESTK    
FGFR1TK    
FGFR2TK    
FGFR3TK    
FGFR4TK    
FGRTK    
FLT4TK    
FRKTK    
FYNTK    
HCKTK    
IGF1RTK    
INSRTK    
INSRRTK    
ITKTK    
JAK2TK    
KDRTK    
LCKTK    
LTKTK    
LYNTK    
MATKTK    
NTRK1TK    
NTRK2TK    
NTRK3TK    
PTK2BTK    
PTK6TK    
RETTK    
SRCTK    
SRMSTK    
SYKTK    
TECTK    
TEKTK    
TNK2TK    
TXKTK    
TYK2TK    
YES1TK    
ZAP70TK    
ACVR1TKL    
ACVR1BTKL    
IRAK1TKL    
IRAK4TKL    
TGFBR1TKL