Kinase profiling results of kinases in KIF 3EIDA_PO5 (CDK2, PDB code: 3EID, chain A)
Template Kinase: CDK2
Template inhibitor: AC1O6YZF

63 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C C C
AKT1AGC   
AKT2AGC   
PDPK1AGC   
PRKCDAGC   
PRKCQAGC   
PKN1AGC   
RPS6KB1AGC   
RPS6KA1AGC   
RPS6KA1CAMK   
CHEK1CAMK   
MARK4CAMK   
NUAK1CAMK   
SIK2CAMK   
STK33CAMK   
STK17ACAMK   
PHKG1CAMK   
PHKG2CAMK   
CDK2CMGC   
CDK4CMGC   
CDK9CMGC   
CSNK2A2CMGC   
CLK1CMGC   
CLK2CMGC   
CLK4CMGC   
DYRK1ACMGC   
DYRK1BCMGC   
DYRK2CMGC   
GSK3BCMGC   
MAPK10CMGC   
MAPK8CMGC   
MAPK9CMGC   
AURKAOther   
AURKBOther   
CAMKK2Other   
PLK1Other   
STK10STE   
MAP2K1STE   
ABL1TK   
ABL2TK   
TNK2TK   
EPHB1TK   
FGFR1TK   
JAK2TK   
JAK3TK   
METTK   
MUSKTK   
FGRTK   
FYNTK   
SRCTK   
YES1TK   
BLKTK   
LCKTK   
LYNTK   
PTK6TK   
ZAP70TK   
ITKTK   
NTRK2TK   
NTRK3TK   
IRAK4TKL   
MAP3K7TKL   
ZAKTKL   

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C C
AKT1AGC     
AKT2AGC     
PDPK1AGC     
PKN1AGC     
PRKCAAGC     
PRKCDAGC     
PRKCQAGC     
RPS6KA1AGC     
RPS6KB1AGC     
CHEK1CAMK     
MARK4CAMK     
NUAK1CAMK     
PHKG1CAMK     
PHKG2CAMK     
SIK2CAMK     
STK17ACAMK     
STK33CAMK     
CDC2CMGC     
CDC2CMGC     
CDK2CMGC     
CDK4CMGC     
CDK6CMGC     
CDK6CMGC     
CDK9CMGC     
CLK1CMGC     
CLK2CMGC     
CLK4CMGC     
CSNK2A2CMGC     
DYRK1ACMGC     
DYRK1BCMGC     
DYRK2CMGC     
GSK3BCMGC     
MAPK10CMGC     
MAPK8CMGC     
MAPK9CMGC     
AURKAOther     
AURKBOther     
CAMKK2Other     
PLK1Other     
MAP2K1STE     
STK10STE     
ABL1TK     
ABL2TK     
BLKTK     
EPHB1TK     
FGFR1TK     
FGRTK     
FYNTK     
ITKTK     
JAK2TK     
JAK3TK     
LCKTK     
LYNTK     
METTK     
MUSKTK     
NTRK2TK     
NTRK3TK     
PTK6TK     
SRCTK     
TNK2TK     
YES1TK     
ZAP70TK     
IRAK4TKL     
MAP3K7TKL     
ZAKTKL