Kinase profiling results of kinases in KIF 3GENA_B43 (BTK, PDB code: 3GEN, chain A)
Template Kinase: BTK
Template inhibitor: 7-Cyclopentyl-5-(4-phenoxy)phenyl-7H-pyrrolo[2,3-d]pyrimidin-4-ylamine

29 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C C C
AKT1AGC   
AURKAOther   
ABL1TK   
TNK2TK   
CSKTK   
EGFRTK   
ERBB2TK   
ERBB4TK   
IGF1RTK   
INSRTK   
KITTK   
PDGFRBTK   
RETTK   
FRKTK   
FGRTK   
FYNTK   
SRCTK   
YES1TK   
BLKTK   
HCKTK   
LCKTK   
LYNTK   
PTK6TK   
SRMSTK   
BMXTK   
BTKTK   
TECTK   
TXKTK   
KDRTK   

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C C
AKT1AGC     
AURKAOther     
ABL1TK     
BLKTK     
BMXTK     
BTKTK     
CSKTK     
EGFRTK     
ERBB2TK     
ERBB4TK     
FGRTK     
FRKTK     
FYNTK     
HCKTK     
IGF1RTK     
INSRTK     
KDRTK     
KITTK     
LCKTK     
LYNTK     
PDGFRBTK     
PTK6TK     
RETTK     
SRCTK     
SRMSTK     
TECTK     
TNK2TK     
TXKTK     
YES1TK