Kinase profiling results of kinases in KIF 2XIKA_J60 (STK25, PDB code: 2XIK, chain A)
Template Kinase: STK25
Template inhibitor: SU11652

59 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C C C C C
GRK1AGC     
GRK4AGC     
GRK7AGC     
PRKCQAGC     
PKN2AGC     
CAMK2ACAMK     
CAMK2DCAMK     
CHEK1CAMK     
DAPK1CAMK     
DAPK2CAMK     
STK17ACAMK     
STK17BCAMK     
MAPKAPK23     
PHKG1CAMK     
PHKG2CAMK     
CDK2CMGC     
CDK5CMGC     
CDKL2CMGC     
DYRK1BCMGC     
DYRK2CMGC     
HIPK1CMGC     
HIPK4CMGC     
GSK3ACMGC     
ICKCMGC     
MAKCMGC     
AURKAOther     
AURKBOther     
AURKCOther     
CAMKK1Other     
CAMKK2Other     
SBK1Other     
PLK2Other     
PAK4STE     
SLKSTE     
MST4STE     
STK24STE     
STK25STE     
TNK1TK     
TNK2TK     
INSRTK     
JAK3TK     
METTK     
MUSKTK     
KITTK     
RETTK     
FGRTK     
FYNTK     
PTK6TK     
ITKTK     
NTRK2TK     
IRAK4TKL     
LRRK2TKL     
MAP3K12TKL     
MAP3K13TKL     
MAP3K11TKL     
MAP3K9TKL     

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C C C
GRK4AGC      
GRK6AGC      
GRK7AGC      
PKN2AGC      
PRKCQAGC      
CAMK2ACAMK      
CAMK2DCAMK      
CHEK1CAMK      
DAPK1CAMK      
DAPK2CAMK      
MAPKAPK2CAMK      
PHKG1CAMK      
PHKG2CAMK      
STK17ACAMK      
CDC2CMGC      
CDC2CMGC      
CDK2CMGC      
CDK5CMGC      
CDK6CMGC      
CDK6CMGC      
DYRK1BCMGC      
DYRK2CMGC      
GSK3ACMGC      
HIPK1CMGC      
HIPK4CMGC      
AURKAOther      
AURKBOther      
AURKCOther      
CAMKK1Other      
CAMKK2Other      
PLK2Other      
MST4STE      
PAK4STE      
SLKSTE      
STK24STE      
STK25STE      
FGRTK      
FYNTK      
INSRTK      
ITKTK      
JAK3TK      
KITTK      
METTK      
MUSKTK      
NTRK2TK      
PTK6TK      
RETTK      
TNK2TK      
IRAK4TKL      
LRRK2TKL      
MAP3K11TKL      
MAP3K9TKL