Kinase profiling results of kinases in KIF 2XRUA_400 (AURKA, PDB code: 2XRU, chain A)
Template Kinase: AURKA
Template inhibitor: VX_680

33 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C C C C C C C C
PDPK1AGC        
PRKACAAGC        
PRKCDAGC        
PRKCQAGC        
CHEK1CAMK        
MAPKAPK23        
CDK2CMGC        
CDK4CMGC        
CDK5CMGC        
CSNK2A1CMGC        
GSK3ACMGC        
GSK3BCMGC        
AURKAOther        
AURKBOther        
AURKCOther        
PLK1Other        
PLK3Other        
MAP4K2STE        
PAK4STE        
ABL1TK        
ALKTK        
EGFRTK        
FGFR1TK        
JAK2TK        
JAK3TK        
RETTK        
LCKTK        
ITKTK        
TXKTK        
TEKTK        
NTRK1TK        

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C C C
PDPK1AGC      
PRKACAAGC      
PRKCDAGC      
PRKCQAGC      
PRKCZAGC      
CHEK1CAMK      
MAPKAPK2CAMK      
CDC2CMGC      
CDC2CMGC      
CDK2CMGC      
CDK4CMGC      
CDK5CMGC      
CSNK2A1CMGC      
GSK3ACMGC      
GSK3BCMGC      
AURKAOther      
AURKBOther      
AURKCOther      
PLK1Other      
PLK3Other      
MAP4K2STE      
PAK4STE      
ABL1TK      
ALKTK      
EGFRTK      
FGFR1TK      
ITKTK      
JAK2TK      
JAK3TK      
LCKTK      
NTRK1TK      
RETTK      
TEKTK      
TXKTK