Kinase profiling results of kinases in KIF 1OIYA_N41 (CDK2, PDB code: 1OIY, chain A)
Template Kinase: CDK2
Template inhibitor: N41

33 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C
ROCK2AGC 
RPS6KA2AGC 
RPS6KA2CAMK 
RPS6KA3AGC 
RPS6KA6AGC 
RPS6KA6CAMK 
NUAK1CAMK 
NUAK2CAMK 
CHEK2CAMK 
TSSK1BCAMK 
CDK2CMGC 
CDK4CMGC 
CSNK2A1CMGC 
CLK2CMGC 
CLK4CMGC 
AURKAOther 
AURKBOther 
AURKCOther 
EIF2AK2Other 
TTKOther 
TNK2TK 
FERTK 
JAK2TK 
JAK3TK 
SRCTK 
YES1TK 
LCKTK 
PTK6TK 
BMXTK 
NTRK3TK 
MAP3K10TKL 
MAP3K11TKL 
MAP3K9TKL 

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C
ROCK2AGC   
RPS6KA2AGC   
RPS6KA3AGC   
RPS6KA6AGC   
CHEK2CAMK   
NUAK1CAMK   
NUAK2CAMK   
TSSK1BCAMK   
CDC2CMGC   
CDC2CMGC   
CDK2CMGC   
CDK4CMGC   
CDK6CMGC   
CDK6CMGC   
CLK2CMGC   
CLK4CMGC   
CSNK2A1CMGC   
AURKAOther   
AURKBOther   
AURKCOther   
TTKOther   
BMXTK   
FERTK   
JAK2TK   
JAK3TK   
LCKTK   
NTRK3TK   
PTK6TK   
SRCTK   
TNK2TK   
YES1TK   
MAP3K10TKL   
MAP3K11TKL   
MAP3K9TKL