Kinase profiling results of kinases in KIF 3MVLA_38P (MAPK14, PDB code: 3MVL, chain A)
Template Kinase: MAPK14
Template inhibitor: 38P

50 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C C C C C C C
GRK7AGC       
PDPK1AGC       
RPS6KA1AGC       
RPS6KA1CAMK       
RPS6KA2AGC       
RPS6KA2CAMK       
RPS6KA6AGC       
RPS6KA6CAMK       
CAMK2DCAMK       
CHEK1CAMK       
HUNKCAMK       
MGC421053       
DAPK1CAMK       
DAPK2CAMK       
DAPK3CAMK       
PHKG2CAMK       
PRKD1CAMK       
PRKD2CAMK       
PRKD3CAMK       
CHEK2CAMK       
CDK2CMGC       
CDK5CMGC       
CSNK2A1CMGC       
CLK2CMGC       
CLK3CMGC       
HIPK1CMGC       
HIPK2CMGC       
HIPK3CMGC       
HIPK4CMGC       
GSK3ACMGC       
GSK3BCMGC       
MAPK1CMGC       
MAPK10CMGC       
MAPK8CMGC       
MAPK9CMGC       
MAPK11CMGC       
MAPK14CMGC       
CHUKOther       
NEK3Other       
NEK2Other       
PLK1Other       
PLK2Other       
PLK3Other       
SLKSTE       
STK10STE       
ABL1TK       
FGFR1TK       
SRCTK       
HCKTK       
LCKTK       
LYNTK       
PTK6TK       

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C C C
GRK7AGC    
PDPK1AGC    
RPS6KA1AGC    
RPS6KA2AGC    
RPS6KA6AGC    
CAMK2DCAMK    
CHEK1CAMK    
CHEK2CAMK    
DAPK1CAMK    
DAPK2CAMK    
DAPK3CAMK    
PHKG2CAMK    
PRKD1CAMK    
PRKD2CAMK    
PRKD3CAMK    
CDC2CMGC    
CDC2CMGC    
CDK2CMGC    
CDK5CMGC    
CLK2CMGC    
CLK3CMGC    
CSNK2A1CMGC    
GSK3ACMGC    
GSK3BCMGC    
HIPK1CMGC    
HIPK2CMGC    
HIPK3CMGC    
HIPK4CMGC    
MAPK1CMGC    
MAPK10CMGC    
MAPK11CMGC    
MAPK14CMGC    
MAPK8CMGC    
MAPK9CMGC    
CHUKOther    
NEK2Other    
NEK3Other    
PLK1Other    
PLK2Other    
PLK3Other    
SLKSTE    
STK10STE    
ABL1TK    
FGFR1TK    
HCKTK    
LCKTK    
LYNTK    
PTK6TK    
SRCTK