Kinase profiling results of kinases in KIF 1R0PA_KSA (MET, PDB code: 1R0P, chain A)
Template Kinase: MET
Template inhibitor: k-252a

28 kinases in the family
Kinase profiling results source
1. Davis et al. Nature Biotechnology.29, 1046-51
2. Anastassiadis, T. et al. Nature Biotechnology.29, 1039-45


Similarity between template inhibitor and test compounds of profiling results

Davis et al.
Nature Biotechnology.29, 1046-51

<1nM    >10uM
KinaseKinase group C
CDK2CMGC 
PCTK2CMGC 
NEK5Other 
NEK2Other 
ALKTK 
LTKTK 
DDR1TK 
EGFRTK 
FERTK 
FESTK 
FGFR1TK 
INSRTK 
JAK1TK 
JAK2TK 
JAK3TK 
METTK 
MUSKTK 
CSF1RTK 
RETTK 
ROS1TK 
NTRK2TK 
NTRK3TK 
FLT4TK 
KDRTK 
TNNI3KTKL 
MAP3K7TKL 
RIPK2TKL 
RIPK4TKL 

Anastassiadis, T. et al.
Nature Biotechnology.29, 1039-45

0%    100%
KinaseKinase group C C
CDK2CMGC  
NEK2Other  
ALKTK  
CSF1RTK  
EGFRTK  
FERTK  
FESTK  
FGFR1TK  
FLT4TK  
INSRTK  
JAK1TK  
JAK2TK  
JAK3TK  
KDRTK  
LTKTK  
METTK  
MUSKTK  
NTRK2TK  
NTRK3TK  
RETTK  
ROS1TK  
MAP3K7TKL  
RIPK2TKL